Target Details
| UniProt AC | P57059 |
|---|---|
| Gene Symbol | SIK1 |
| Protein Name | Serine/threonine-protein kinase SIK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 192
- Clinical molecules 11
- Avg pChEMBL 7.69
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (192)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AWLHPMOLJAWKDL
|
10.0 | IC50 | 3 | — | |
KDPXVKRYHKSBPY
|
10.0 | IC50 | 3 | — | |
WXCYMIOQVROELY
|
10.0 | IC50 | 3 | — | |
DYMFNPBLDKXKJA
|
9.7 | IC50 | 3 | — | |
XHPICGSLCSAZKX
|
9.7 | IC50 | 3 | — | |
HSQLWSUNRMTGGO
|
9.4 | IC50 | 3 | — | |
YATIMLFNGFQTCA
|
9.4 | IC50 | 3 | — | |
WMCHGBLGKMZDJD
|
9.3 | IC50 | 3 | — | |
YMSJZKSIBUPNHN
|
9.3 | IC50 | 3 | — | |
VATIVDMNNPRBCN
|
9.2 | IC50 | 3 | — | |
YCOQHBLWDSAZRB
|
9.2 | IC50 | 3 | — | |
CAJPKOHOPAWXRV
|
9.2 | IC50 | 3 | — | |
LTQKUGJNXFIXKC
|
9.1 | IC50 | 3 | — | |
AQXQPESYCSEOOG
|
9.1 | IC50 | 3 | — | |
BQKJBKRZMBOHNT
|
9.1 | IC50 | 3 | — | |
MXNBWDNCIZQCIL
|
9.1 | IC50 | 3 | — | |
BIYKGGOFJOFQIZ
|
9.1 | IC50 | 3 | — | |
LYSXGFLZKDKZDF
|
9.1 | IC50 | 3 | — | |
BIYKGGOFJOFQIZ
|
9.0 | IC50 | 3 | — | |
HOKRUYIIDRQYFK
|
8.9 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.9 | IC50 | 408 | — | |
UEQMHAFWQDRPMU
|
8.9 | IC50 | 3 | — | |
INXQKXZSUNICKV
|
8.8 | IC50 | 3 | — | |
YOWQNRVRQMOXAT
|
8.8 | IC50 | 3 | — | |
FQZGWTSGSBKLBT
|
8.8 | IC50 | 3 | — | |
OKSHQZCQVDERIF
|
8.8 | IC50 | 3 | — | |
PNAUGSWMKOHDJF
|
8.8 | IC50 | 3 | — | |
FGLQSISJARINNB
|
8.7 | IC50 | 3 | — | |
PFTXFNSHFZLJNT
|
8.7 | IC50 | 17 | — | |
WDNAXOPVZIEECR
|
8.7 | IC50 | 11 | — | |
QVUYJTWSZWCKHP
|
8.7 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.7 | Kd | 213 | — | |
AWVUPXUQWGNTHF
|
8.6 | IC50 | 3 | — | |
CFNFPVIKPAPVOV
|
8.6 | IC50 | 3 | — | |
RPDJXKWOAHHTBX
|
8.6 | IC50 | 3 | — | |
OMDTWHBLOYOZGL
|
8.6 | IC50 | 3 | — | |
QBSNPDJXAMBWIZ
|
8.6 | IC50 | 3 | — | |
XCGUGTWHQADPNS
|
8.6 | IC50 | 3 | — | |
AQXQPESYCSEOOG
|
8.6 | IC50 | 3 | — | |
HSYDEPQAUCZNGP
|
8.6 | IC50 | 3 | — | |
JVBRZBKYIRZVJE
|
8.6 | IC50 | 3 | — | |
SVNQOEFGBNGPSZ
|
8.6 | IC50 | 3 | — | |
WKZOFECSVXLTOB
|
8.6 | IC50 | 3 | — | |
NDNNIKHUOLIORS
|
8.5 | IC50 | 3 | — | |
NXSJMRCTGYTSTK
|
8.5 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
8.5 | Kd | 170 | — | |
VFDIZCUBJRZYFL
|
8.5 | IC50 | 3 | — | |
DNKJWTDFPIZFNK
|
8.5 | IC50 | 3 | — | |
QOOLIAIGEONMHK
|
8.5 | IC50 | 3 | — | |
RZXPVLRGCBTJSU
|
8.4 | IC50 | 3 | — |