Target Details
| UniProt AC | P57058 |
|---|---|
| Gene Symbol | HUNK |
| Protein Name | Hormonally up-regulated neu tumor-associated kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 11
- Clinical molecules 5
- Avg pChEMBL 6.45
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CTNPALGJUAXMMC
|
8.4 | Kd | 151 | — | |
BMGQWWVMWDBQGC
|
6.6 | Kd | 147 | Yes | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
PIQCTGMSNWUMAF
|
6.4 | Kd | 137 | Yes | |
YYLKKYCXAOBSRM
|
6.3 | Kd | 191 | — | |
WINHZLLDWRZWRT
|
6.3 | Kd | 201 | Yes | |
UIARLYUEJFELEN
|
6.2 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
6.2 | Kd | 408 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |