Target Details
| UniProt AC | P56817 |
|---|---|
| Gene Symbol | BACE1 |
| Protein Name | Beta-secretase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00026 (Asp) |
Summary
- Multi-target molecules 3,050
- Clinical molecules 3
- Avg pChEMBL 7.76
KEGG Pathways (1)
Active Molecules (3,050)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEENGVHYCRGRAD
|
9.0 | Ki | 2 | — | |
SSCPZMVDBVQQMX
|
9.0 | Ki | 2 | — | |
UIRBVORWZZIYQQ
|
9.0 | IC50 | 2 | — | |
UOHXUSCZQJMWQO
|
9.0 | IC50 | 2 | — | |
VDXQVJAEEQGQLD
|
9.0 | Ki | 2 | — | |
VKZQOAUIZVISCN
|
9.0 | Ki | 2 | — | |
VQYBNNOSTNVFEJ
|
9.0 | IC50 | 2 | — | |
WPFPYTKQXHYXQI
|
9.0 | Ki | 2 | — | |
WTKQJNKMIICWFI
|
9.0 | IC50 | 2 | — | |
ZDBCSCLTQTZDDK
|
9.0 | IC50 | 2 | — | |
ZJIPAWSHYBXAKX
|
9.0 | IC50 | 2 | — | |
ZKRIRTXSSDEWSN
|
9.0 | Ki | 2 | — | |
ZRQWZDZYZAYTLY
|
9.0 | Ki | 2 | — | |
ISZZSQRCJWJMMV
|
9.0 | IC50 | 2 | — | |
OTSGTAACGWFXCL
|
9.0 | IC50 | 2 | — | |
FVAIYSHJXOSXKA
|
9.0 | IC50 | 2 | — | |
MTGMNKBRNQNEFJ
|
9.0 | IC50 | 2 | — | |
QGPBROSNFKNVFL
|
9.0 | Ki | 2 | — | |
UZVDKSGFSMHFCE
|
9.0 | IC50 | 2 | — | |
DZESCCQYAGJZKL
|
9.0 | IC50 | 2 | — | |
JLFSIOZYUYAVER
|
9.0 | IC50 | 2 | — | |
JTCINPNYZFDZEO
|
9.0 | IC50 | 2 | — | |
QZZQLTNGTRLGGZ
|
9.0 | IC50 | 2 | — | |
BJOCXJJVELLFKM
|
9.0 | Ki | 3 | — | |
LWCYPSYNLAAESS
|
9.0 | IC50 | 2 | — | |
OBVOAGZBBSFJLL
|
9.0 | IC50 | 2 | — | |
PERQGBHIWDTVOX
|
9.0 | IC50 | 2 | — | |
SQYPMCICTARIJE
|
9.0 | IC50 | 2 | — | |
VJNUVDOJKFVXPP
|
9.0 | Ki | 2 | — | |
BIPOCRRWZJCZAC
|
8.9 | IC50 | 2 | — | |
DJDZRLDHUXKNCV
|
8.9 | IC50 | 2 | — | |
YQLVXTJTQKINJB
|
8.9 | IC50 | 2 | — | |
AXBMNVOPTJGHDS
|
8.9 | IC50 | 2 | — | |
BCPJXJSUDZCZSL
|
8.9 | IC50 | 2 | — | |
HKNVQAYILMKLSZ
|
8.9 | IC50 | 2 | — | |
MFNGXEDOZQICAD
|
8.9 | IC50 | 2 | — | |
QRKJDOAKSMDBOV
|
8.9 | IC50 | 2 | — | |
QUCBIFARZXBMHU
|
8.9 | IC50 | 2 | — | |
XZUSTFQBDGMJHQ
|
8.9 | IC50 | 2 | — | |
YBKXIEMWSKQLOV
|
8.9 | IC50 | 2 | — | |
AZSIDVKSWAWKLB
|
8.9 | IC50 | 2 | — | |
HYFDUAZKGHOXSC
|
8.9 | IC50 | 2 | — | |
CFIWWTUUSMMDDA
|
8.9 | Ki | 2 | — | |
DOTNQRHMAHZRQZ
|
8.9 | IC50 | 2 | — | |
GAZOPRYFZALSHV
|
8.9 | Ki | 2 | — | |
GSXNFTYLLVDBEE
|
8.9 | Ki | 2 | — | |
HLUAIMQRMMIEHR
|
8.9 | Ki | 2 | — | |
KAUGEXWMBITOIF
|
8.9 | IC50 | 2 | — | |
LPXQIVMHUYETDK
|
8.9 | IC50 | 2 | — | |
NRIZDKUKBXCEHA
|
8.9 | IC50 | 2 | — |