Target Details
| UniProt AC | P56817 |
|---|---|
| Gene Symbol | BACE1 |
| Protein Name | Beta-secretase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00026 (Asp) |
Summary
- Multi-target molecules 3,050
- Clinical molecules 3
- Avg pChEMBL 7.76
KEGG Pathways (1)
Active Molecules (3,050)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KIEWLGRGIVAZSL
|
8.7 | IC50 | 2 | — | |
MIHYIRSACAPCTC
|
8.7 | IC50 | 2 | — | |
MQSSLRBZFVPDKD
|
8.7 | IC50 | 2 | — | |
NXJUOWRPEGSDFT
|
8.7 | IC50 | 2 | — | |
OGEVSLFGHQATOX
|
8.7 | Ki | 2 | — | |
OUXYSMGAVPZBDV
|
8.7 | IC50 | 2 | — | |
PKBZVGSMKHULBV
|
8.7 | IC50 | 2 | — | |
SIQCBZMRMXEYSX
|
8.7 | IC50 | 2 | — | |
SUGIUUXWIMLLJY
|
8.7 | IC50 | 2 | — | |
VPVXNJPVCHXXDB
|
8.7 | Ki | 2 | — | |
WVWGFCSJXQRWQR
|
8.7 | Ki | 2 | — | |
WYHSXLPYCWHUCK
|
8.7 | IC50 | 2 | — | |
CFESCKXVBKHVFX
|
8.7 | IC50 | 2 | — | |
CTDUMLUKUOGMRV
|
8.7 | IC50 | 2 | — | |
MTNHQSSEAULFMW
|
8.7 | IC50 | 2 | — | |
OTEJLQDKYJIXPC
|
8.7 | IC50 | 2 | — | |
BLPDQFTZIQGBQQ
|
8.7 | Ki | 2 | — | |
CHZHWZAKWGFQNL
|
8.7 | IC50 | 4 | — | |
JZALFYMKSGBBQK
|
8.7 | Ki | 2 | — | |
KJHZTBSKBYEHQO
|
8.7 | IC50 | 2 | — | |
SJWYDDZFJMFIGS
|
8.7 | Ki | 2 | — | |
SKNSXIIPICYXKY
|
8.7 | IC50 | 2 | — | |
WKDNQONLGXOZRG
|
8.7 | IC50 | 2 | — | |
XTQZDTBINKMEKZ
|
8.7 | IC50 | 2 | — | |
YHYKUSGACIYRML
|
8.7 | Ki | 2 | — | |
KJFQHLLASMWVFN
|
8.7 | IC50 | 2 | — | |
NNIPUJZFEKQESE
|
8.7 | IC50 | 2 | — | |
PQEHEWHVXPCYGP
|
8.7 | IC50 | 2 | — | |
UULZRQYJOWPKGT
|
8.7 | IC50 | 2 | — | |
VFRMWJSJMHBDCM
|
8.7 | Ki | 2 | — | |
ZFKNVJXLEJYKRB
|
8.7 | IC50 | 2 | — | |
BHCDFMZEDWIROP
|
8.6 | IC50 | 2 | — | |
IJKMXPBVUFGDLK
|
8.6 | Ki | 2 | — | |
JBARGSXIUKTHNW
|
8.6 | IC50 | 2 | — | |
JWLYVBNCRPQOOA
|
8.6 | IC50 | 2 | — | |
OYVJXWZSTBCONR
|
8.6 | IC50 | 2 | — | |
PCEGZDCSGKYRGF
|
8.6 | IC50 | 2 | — | |
QLVXMZONSZVPIM
|
8.6 | Ki | 2 | — | |
QQHWYFAIJDVZQX
|
8.6 | IC50 | 2 | — | |
RZKUSOMDXZAIJY
|
8.6 | Ki | 2 | — | |
SCKAYIQTMXSRCI
|
8.6 | IC50 | 2 | — | |
WBFTZCDXILITBE
|
8.6 | IC50 | 2 | — | |
XSPYGYYSPGDIRH
|
8.6 | IC50 | 2 | — | |
ZXRHVPQEUUVSBF
|
8.6 | IC50 | 2 | — | |
AGPHPRAMUFTZTL
|
8.6 | IC50 | 2 | — | |
GKJLWBZUMCCOIW
|
8.6 | IC50 | 2 | — | |
SECXNYKABFAMCL
|
8.6 | IC50 | 2 | — | |
CQQMWBPWYUPVOC
|
8.6 | IC50 | 4 | — | |
DDHXRMBHBIIYGG
|
8.6 | IC50 | 2 | — | |
DHESWQSXKSVRPU
|
8.6 | IC50 | 2 | — |