Target Details
| UniProt AC | P56817 |
|---|---|
| Gene Symbol | BACE1 |
| Protein Name | Beta-secretase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00026 (Asp) |
Summary
- Multi-target molecules 3,050
- Clinical molecules 3
- Avg pChEMBL 7.76
KEGG Pathways (1)
Active Molecules (3,050)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ANDKFLRZHHHXMI
|
10.2 | IC50 | 2 | — | |
CHFWFILSMSLUCS
|
10.2 | IC50 | 2 | — | |
JSBFBQWKNPPENK
|
10.1 | IC50 | 2 | — | |
SUUZEAQMBKCXPP
|
10.0 | IC50 | 2 | — | |
RSXKHMYUKFBRTL
|
10.0 | IC50 | 2 | — | |
UDROXIDKAFGJQP
|
9.9 | Ki | 3 | — | |
UZFAOTIMARRSKT
|
9.9 | IC50 | 2 | — | |
AKFBRKWOFKXXKV
|
9.8 | IC50 | 2 | — | |
AOKIPVSNIFDFTR
|
9.8 | IC50 | 2 | — | |
FSZBZCCCGRRZMK
|
9.8 | IC50 | 2 | — | |
HENFIGCJZYPGHN
|
9.7 | IC50 | 2 | — | |
IPUJINDWAGRAHN
|
9.7 | IC50 | 2 | — | |
WNOKZFQDOPPTQP
|
9.7 | IC50 | 2 | — | |
BKSJVUKEEUFBSI
|
9.7 | IC50 | 2 | — | |
JZRRLACUGZNGSR
|
9.7 | IC50 | 2 | — | |
UYXLCQKZJUELFM
|
9.7 | IC50 | 2 | — | |
LNCNDCQMCRPPAO
|
9.7 | IC50 | 2 | — | |
GJKNFCVMUNZMOD
|
9.7 | IC50 | 2 | — | |
NURKHPHCXJUBHN
|
9.6 | IC50 | 2 | — | |
URYGNWAQODMINB
|
9.6 | IC50 | 2 | — | |
ULUVFLUZTKOQFK
|
9.6 | IC50 | 2 | — | |
WZMUQDQOZDDLLR
|
9.6 | IC50 | 2 | — | |
GUFJTLQVFGVMAQ
|
9.6 | Ki | 3 | — | |
KSQXUTYVDJUGIQ
|
9.6 | IC50 | 2 | — | |
BQXOCDCEKQYJHJ
|
9.6 | IC50 | 2 | — | |
LXTSXUJESINVNI
|
9.6 | IC50 | 2 | — | |
ONSHBIJSSOXNFW
|
9.6 | IC50 | 2 | — | |
UUXDVXFJLGMTAM
|
9.6 | IC50 | 2 | — | |
ZOGJTGSYBFRPTG
|
9.6 | IC50 | 2 | — | |
KDARIEFFIVBDRF
|
9.6 | IC50 | 2 | — | |
AAWPKTSUNVJJFB
|
9.5 | IC50 | 2 | — | |
JJADJMODPHLYCB
|
9.5 | IC50 | 2 | — | |
NSMFFDBQMBKGNX
|
9.5 | IC50 | 2 | — | |
IOGNYIFQSZMVPU
|
9.5 | IC50 | 2 | — | |
SRIRNELXGCWCRJ
|
9.5 | IC50 | 2 | — | |
XCVCPWYOVVQNJH
|
9.5 | IC50 | 2 | — | |
ASNUKCLRXVDLSX
|
9.5 | IC50 | 2 | — | |
DRRNRXVQVQEOLP
|
9.5 | IC50 | 2 | — | |
OFAZWNGNAATRSH
|
9.5 | Ki | 3 | — | |
PENUXFUKWLPNBH
|
9.5 | IC50 | 2 | — | |
BOVNRMGLJLBYEO
|
9.5 | IC50 | 2 | — | |
GZYRQCRYXGTKID
|
9.5 | IC50 | 2 | — | |
KGEBCNTYUXGVQW
|
9.5 | IC50 | 2 | — | |
OOLVBHNAPKNWGY
|
9.5 | IC50 | 2 | — | |
UJTLXAIVCCJWHY
|
9.5 | IC50 | 2 | — | |
YZZCVUIDSNUXDI
|
9.5 | IC50 | 2 | — | |
MPLHANQZLPTTKT
|
9.5 | IC50 | 2 | — | |
PHHUTLNIMVWRRK
|
9.5 | IC50 | 2 | — | |
YIQUYGRGOCRWFL
|
9.5 | IC50 | 2 | — | |
LNCNDCQMCRPPAO
|
9.5 | IC50 | 2 | — |