Target Details
| UniProt AC | P56373 |
|---|---|
| Gene Symbol | P2RX3 |
| Protein Name | P2X purinoceptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00864 (P2X_receptor) |
Summary
- Multi-target molecules 550
- Clinical molecules 0
- Avg pChEMBL 7.46
KEGG Pathways (4)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KKCKQAQSHHVSCO
|
7.1 | IC50 | 2 | — | |
PFTSILFRTYLFOO
|
7.1 | IC50 | 2 | — | |
CUYVVUGLFUIZAZ
|
7.1 | IC50 | 3 | — | |
DUSNKKLMFUTVFU
|
7.1 | IC50 | 2 | — | |
NWTVSPCFEGLAFO
|
7.1 | IC50 | 2 | — | |
XNMZCBBYALDDDV
|
7.1 | Ki | 2 | — | |
ZBRXLMDGZXDHGV
|
7.1 | IC50 | 2 | — | |
MPEWWUPGWDTWHF
|
7.1 | IC50 | 2 | — | |
SHLRNWXFYHGFLL
|
7.1 | IC50 | 2 | — | |
BXYCNACOQSAWFQ
|
7.0 | Ki | 2 | — | |
SNULHIJATIOARQ
|
7.0 | Ki | 2 | — | |
KYDLIDYIDLJOAK
|
7.0 | IC50 | 2 | — | |
DRAPDSWDHFUIHZ
|
7.0 | Ki | 2 | — | |
LAKQJAHJFOBGJH
|
7.0 | IC50 | 2 | — | |
MOJZESVRLRZYMR
|
7.0 | IC50 | 2 | — | |
DRKKSNGJFWQKKN
|
7.0 | IC50 | 2 | — | |
LLNHATOQNPRUDF
|
7.0 | IC50 | 2 | — | |
ACBYIIVYPXEGQW
|
7.0 | IC50 | 2 | — | |
ZBNNSVNQQSLELF
|
7.0 | IC50 | 2 | — | |
DFGOJQUEWDGMKI
|
7.0 | IC50 | 2 | — | |
FVGXVLFIHFQXPP
|
7.0 | IC50 | 2 | — | |
HGARQXXUVFFGNI
|
7.0 | IC50 | 2 | — | |
SEUOQQWVKWQBQA
|
7.0 | IC50 | 2 | — | |
MWBSFWZECXCRJX
|
7.0 | IC50 | 2 | — | |
NTNQBRZBMXLLSB
|
7.0 | IC50 | 2 | — | |
XDSMVWUQPSBETH
|
7.0 | Ki | 2 | — | |
USOMQOKPGJTCRC
|
7.0 | IC50 | 2 | — | |
YEZMTVSPNRFAKT
|
7.0 | IC50 | 2 | — | |
NLLVDMMXBRFWGS
|
7.0 | IC50 | 2 | — | |
ULSBLOPPTNALIT
|
7.0 | IC50 | 2 | — | |
WWWCBSCSEOPHLV
|
7.0 | IC50 | 2 | — | |
XUTUDMYKUNRZSS
|
7.0 | Ki | 2 | — | |
HVLSFPXITWENER
|
6.9 | IC50 | 2 | — | |
ACKCNQSPIBKCRO
|
6.9 | Ki | 2 | — | |
DRTIWPFAAYZULE
|
6.9 | IC50 | 2 | — | |
GBDWWYIZWHGLEN
|
6.9 | IC50 | 2 | — | |
LILYTSLDQVOVAO
|
6.9 | Ki | 2 | — | |
QAFMSMLCHQICCA
|
6.9 | Ki | 2 | — | |
VMBJAODLXQLQDW
|
6.9 | Ki | 2 | — | |
MJOIQVQXAGARNV
|
6.9 | Ki | 2 | — | |
SHLRNWXFYHGFLL
|
6.9 | IC50 | 2 | — | |
OHKYSCNGLWLOFA
|
6.9 | IC50 | 2 | — | |
VUXDKUAYZMWTBM
|
6.9 | IC50 | 2 | — | |
XPCVTIPTPXJKOD
|
6.9 | IC50 | 2 | — | |
ZUDOFWCYSIYMFD
|
6.9 | Ki | 2 | — | |
PZARJLLATJAKMG
|
6.9 | IC50 | 2 | — | |
QVZLKMLKJOKUHQ
|
6.9 | IC50 | 2 | — | |
OMDXBHIZMDEQDL
|
6.9 | IC50 | 2 | — | |
FRKYVICUHIHNMI
|
6.8 | Ki | 2 | — | |
FJEGDSNOOKRLRP
|
6.8 | IC50 | 2 | — |