Target Details
| UniProt AC | P56373 |
|---|---|
| Gene Symbol | P2RX3 |
| Protein Name | P2X purinoceptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00864 (P2X_receptor) |
Summary
- Multi-target molecules 550
- Clinical molecules 0
- Avg pChEMBL 7.46
KEGG Pathways (4)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZERBIURYMMOJBU
|
7.5 | IC50 | 2 | — | |
LBHYSUNETNFKQT
|
7.5 | Ki | 2 | — | |
IVUVTQZOIPAQFU
|
7.4 | IC50 | 2 | — | |
KGDPEGCMVCXNPY
|
7.4 | IC50 | 2 | — | |
MPEWWUPGWDTWHF
|
7.4 | IC50 | 2 | — | |
QGKWEGPZHJOINP
|
7.4 | Ki | 2 | — | |
QOJBRGRPZKZVKC
|
7.4 | IC50 | 2 | — | |
KGDPEGCMVCXNPY
|
7.4 | IC50 | 2 | — | |
KTFAMKPHNDUKLL
|
7.4 | IC50 | 2 | — | |
LZHFVMNPYNSOFI
|
7.4 | Ki | 2 | — | |
NXXXMKXJEBTPJP
|
7.4 | Ki | 2 | — | |
PXQNUEJJIJCDAS
|
7.4 | Ki | 2 | — | |
RCAMJYBTCSWONV
|
7.4 | IC50 | 2 | — | |
RXZNFBASJKIFOC
|
7.4 | IC50 | 2 | — | |
WJNIKDPPMLYZOS
|
7.4 | IC50 | 2 | — | |
JJXMVDHMQZPOJY
|
7.4 | IC50 | 2 | — | |
AAAAEENPAALFRN
|
7.4 | IC50 | 2 | — | |
GGWJLMLTKXSELO
|
7.4 | IC50 | 2 | — | |
MLKRPMMAEMGGNI
|
7.4 | IC50 | 2 | — | |
UVADKIPIQNNHRJ
|
7.4 | IC50 | 2 | — | |
JZRSBKDBMGCFDH
|
7.4 | IC50 | 2 | — | |
NLTUCYMLOPLUHL
|
7.4 | Ki | 2 | — | |
PQZKBUDIGDWISA
|
7.4 | IC50 | 2 | — | |
NMFJPJCALUOMRM
|
7.4 | IC50 | 2 | — | |
OVUBAZICSOPILB
|
7.4 | IC50 | 2 | — | |
KTZHJRKMBNLACT
|
7.4 | IC50 | 2 | — | |
QNHMPCGUVCJNLG
|
7.4 | IC50 | 2 | — | |
COCLYUAEQYUAPW
|
7.4 | IC50 | 2 | — | |
FPSSQFUABOQNNZ
|
7.4 | IC50 | 2 | — | |
GFPCDVNWJYDKRC
|
7.4 | Ki | 2 | — | |
KVPJWYRZJZEFAA
|
7.4 | IC50 | 2 | — | |
UKVBYTFAVWLLPI
|
7.4 | IC50 | 2 | — | |
VBGYUQHZGFCORX
|
7.4 | IC50 | 2 | — | |
BHRXSWOPMLFOCG
|
7.3 | IC50 | 2 | — | |
GKNCXHRLEQHNKW
|
7.3 | IC50 | 2 | — | |
GOFUMWOIVIXXIJ
|
7.3 | IC50 | 2 | — | |
HLWURFKMDLAKOD
|
7.3 | IC50 | 2 | — | |
KRMAXJMLJAVOGJ
|
7.3 | IC50 | 2 | — | |
OSQFXHWKOIFZOO
|
7.3 | Ki | 2 | — | |
YTKWIWSPGJOVJL
|
7.3 | IC50 | 2 | — | |
CAKLWYTTWVXMCY
|
7.3 | IC50 | 2 | — | |
JWRPHAGJMIAQMD
|
7.3 | IC50 | 2 | — | |
LHUVAVZJRUVQTK
|
7.3 | IC50 | 2 | — | |
OQZFQIHVHFJDIX
|
7.3 | IC50 | 2 | — | |
COCLYUAEQYUAPW
|
7.3 | IC50 | 2 | — | |
NLIHPCYXRYQPSD
|
7.3 | Ki | 2 | — | |
CFTQNAYGOFQJGD
|
7.3 | IC50 | 2 | — | |
CTSWGKHAONRRHA
|
7.3 | IC50 | 2 | — | |
GKNCXHRLEQHNKW
|
7.3 | IC50 | 2 | — | |
JVDBFDLYRVYCCM
|
7.3 | Ki | 2 | — |