Target Details
| UniProt AC | P56373 |
|---|---|
| Gene Symbol | P2RX3 |
| Protein Name | P2X purinoceptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00864 (P2X_receptor) |
Summary
- Multi-target molecules 550
- Clinical molecules 0
- Avg pChEMBL 7.46
KEGG Pathways (4)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UMZMQINYOLOMAX
|
6.5 | IC50 | 2 | — | |
UXZIOQCGIFBABV
|
6.5 | IC50 | 2 | — | |
XRCWMLVPRKTAQG
|
6.5 | IC50 | 2 | — | |
WCOLFQGIJSKNOR
|
6.5 | Ki | 2 | — | |
BYVUBCIRZIXXCV
|
6.5 | IC50 | 2 | — | |
UDVIAMRWOLIUAE
|
6.5 | IC50 | 3 | — | |
BPRNAIIYYOQQKN
|
6.4 | IC50 | 2 | — | |
UFZTZBNSLXELAL
|
6.4 | Ki | 2 | — | |
DOIRBVVZCMJEJL
|
6.4 | IC50 | 2 | — | |
DUWZFANLTWXYCX
|
6.4 | IC50 | 2 | — | |
HIKYTWIVLKHYIM
|
6.4 | IC50 | 2 | — | |
IBCZHROKDLOJJF
|
6.4 | IC50 | 2 | — | |
IKPGHRSYEVJPTH
|
6.4 | Ki | 2 | — | |
IQEIDXMZRHBDKY
|
6.4 | IC50 | 2 | — | |
OAKPWEUQDVLTCN
|
6.4 | Ki | 4 | — | |
BEWVSTIRWSWSRV
|
6.4 | IC50 | 2 | — | |
IUVDXBRGFXCMBT
|
6.4 | IC50 | 2 | — | |
PEMLUSSWDFVTHU
|
6.4 | IC50 | 2 | — | |
WRJITTKUXGEQBF
|
6.4 | IC50 | 3 | — | |
IDGSUOPUMKFOSU
|
6.3 | Ki | 2 | — | |
JEFRBKGYXHTEFD
|
6.3 | Ki | 2 | — | |
XTWYTFMLZFPYCI
|
6.3 | Ki | 6 | — | |
OSQOURHXWJQPNS
|
6.3 | IC50 | 2 | — | |
GPAJMPPOAYJSIV
|
6.3 | IC50 | 2 | — | |
AFYIVHVQSPKIIO
|
6.3 | IC50 | 2 | — | |
BKQZGVPRPNNNDW
|
6.3 | IC50 | 2 | — | |
MMVNDZWNOYKPLL
|
6.2 | Ki | 2 | — | |
MPNBZJLDZOIHAR
|
6.2 | Ki | 2 | — | |
FJEGDSNOOKRLRP
|
6.2 | IC50 | 2 | — | |
HNBMXRXUZXPWRO
|
6.2 | Ki | 2 | — | |
NTIPPLUXKZVJHM
|
6.2 | IC50 | 2 | — | |
BMGSNGSJUJYWRK
|
6.2 | IC50 | 2 | — | |
LHUYOPDVSCBYGR
|
6.2 | IC50 | 2 | — | |
QWGYVISNASORKE
|
6.2 | IC50 | 2 | — | |
AKHUMVIUALSLOB
|
6.2 | IC50 | 2 | — | |
TYZFKVQYKKYAAW
|
6.2 | Ki | 2 | — | |
QQLWOWLPRQTDCM
|
6.2 | IC50 | 2 | — | |
JYDDCTCHITXHNX
|
6.2 | Ki | 2 | — | |
LDLJTALPLRVDBD
|
6.2 | IC50 | 2 | — | |
XDHNQDDQEHDUTM
|
6.1 | IC50 | 2 | — | |
HZABZKYZDQPWMV
|
6.1 | IC50 | 2 | — | |
MPEWWUPGWDTWHF
|
6.1 | IC50 | 2 | — | |
OLLXXVGRMYIESK
|
6.1 | IC50 | 2 | — | |
JQUVQWMHZSYCRQ
|
6.1 | IC50 | 2 | — | |
SJEKZQLZHAPABT
|
6.1 | IC50 | 2 | — | |
MUCFYQFETABRSU
|
6.0 | IC50 | 2 | — | |
MNDBFJPWTMCRLX
|
6.0 | Ki | 2 | — | |
OUQUOVKPHMOXRY
|
6.0 | IC50 | 2 | — | |
QIUGFNUDQJFIFZ
|
6.0 | IC50 | 2 | — | |
YSCNMFDFYJUPEF
|
6.0 | IC50 | 2 | — |