Target Details
| UniProt AC | P56199 |
|---|---|
| Gene Symbol | ITGA1 |
| Protein Name | Integrin alpha-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00092 (VWA) |
Summary
- Multi-target molecules 6
- Clinical molecules 0
- Avg pChEMBL 7.04
KEGG Pathways (11)
- Arrhythmogenic right ventricular cardiomyopathy
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NVVGCQABIHSJSQ
|
8.2 | IC50 | 6 | — | |
XXVHVXVVXGOJQZ
|
7.5 | IC50 | 4 | — | |
FXYDXLJEJBXFBD
|
7.3 | IC50 | 5 | — | |
FXYDXLJEJBXFBD
|
7.1 | IC50 | 6 | — | |
FXYDXLJEJBXFBD
|
6.2 | IC50 | 7 | — | |
FXYDXLJEJBXFBD
|
6.0 | IC50 | 6 | — |