Target Details
| UniProt AC | P55210 |
|---|---|
| Gene Symbol | CASP7 |
| Protein Name | Caspase-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 306
- Clinical molecules 0
- Avg pChEMBL 7.38
KEGG Pathways (14)
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Legionellosis
- Lipid and atherosclerosis
- Non-alcoholic fatty liver disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Salmonella infection
- TNF signaling pathway
Active Molecules (306)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PBRJUWKZXWXZNB
|
6.7 | IC50 | 2 | — | |
ZQDAIIUFJKGWON
|
6.7 | IC50 | 2 | — | |
CXBBLGYLOAZXJT
|
6.7 | IC50 | 5 | — | |
IVNMNOZULIYBTB
|
6.7 | IC50 | 2 | — | |
ONFHORMKUAUOAQ
|
6.7 | IC50 | 2 | — | |
HCWVNDBXTZOJJT
|
6.6 | IC50 | 2 | — | |
HOUWXSCEZSJNPK
|
6.6 | IC50 | 2 | — | |
JLXZUACSFOZXOH
|
6.6 | IC50 | 2 | — | |
YDWMZYBWKLFQKO
|
6.6 | IC50 | 3 | — | |
MIRPJNSLZMOWQE
|
6.6 | IC50 | 2 | — | |
RBCPNDRFXKBOQT
|
6.6 | IC50 | 2 | — | |
SGVNFLQYMIJSSK
|
6.6 | IC50 | 3 | — | |
RQWMOUMJTFUKRW
|
6.5 | IC50 | 2 | — | |
VGTVMULINBNZTO
|
6.5 | IC50 | 2 | — | |
VIUJQQJJJZNKDP
|
6.5 | IC50 | 4 | — | |
JPTDPTOWOMFBRY
|
6.5 | Ki | 2 | — | |
MEOSEAYZHVITJF
|
6.5 | IC50 | 3 | — | |
MEOSEAYZHVITJF
|
6.5 | IC50 | 3 | — | |
APKUVGMUIXJJAR
|
6.5 | IC50 | 2 | — | |
PAPREHNJYFBQSL
|
6.5 | IC50 | 2 | — | |
QKVWMYQCBWNCQH
|
6.5 | IC50 | 2 | — | |
SMINLRKVPPXJGK
|
6.5 | IC50 | 2 | — | |
NVUAKKWTWHVSEV
|
6.5 | IC50 | 2 | — | |
FOGVBUNJXCEAOT
|
6.5 | IC50 | 2 | — | |
AYNCKCVIBWBSLQ
|
6.5 | IC50 | 2 | — | |
FATMLWUGEBQNST
|
6.4 | IC50 | 2 | — | |
NQNOSUGXDKSHRE
|
6.4 | IC50 | 3 | — | |
ULYGADBUPXIMGK
|
6.4 | IC50 | 2 | — | |
QGZFJAMNGXQLQV
|
6.4 | IC50 | 2 | — | |
QIAVLJUPQMHWEU
|
6.4 | IC50 | 2 | — | |
YIOFGHHAURBGSJ
|
6.4 | IC50 | 3 | — | |
FZAVLWDWOZHIBJ
|
6.4 | IC50 | 3 | — | |
MFHQDLHNUMVDLA
|
6.4 | IC50 | 4 | — | |
IRBBDJYBNHNLKO
|
6.4 | IC50 | 2 | — | |
VBLKIMKAYGBRKC
|
6.3 | IC50 | 2 | — | |
FMTZTJFXNZOBIQ
|
6.3 | Ki | 5 | — | |
IPHOHJYEJYKOEY
|
6.3 | IC50 | 2 | — | |
RGINHWLPKMMZFM
|
6.3 | IC50 | 3 | — | |
RGINHWLPKMMZFM
|
6.3 | IC50 | 3 | — | |
VOOBNDVVTJIXRQ
|
6.3 | IC50 | 2 | — | |
YYHQMSJBLNLPNZ
|
6.3 | IC50 | 2 | — | |
HOONNWPQCPKYFI
|
6.3 | IC50 | 2 | — | |
HWKXAKRQXXUBFD
|
6.3 | IC50 | 3 | — | |
HWKXAKRQXXUBFD
|
6.3 | IC50 | 3 | — | |
NLZNSSWGRVBWIX
|
6.2 | IC50 | 4 | — | |
CLKQXEGDLZQTME
|
6.2 | IC50 | 4 | — | |
NMZRNLRSVKUVJC
|
6.2 | IC50 | 2 | — | |
QIOIIQRMCCDEQM
|
6.2 | IC50 | 2 | — | |
NHIDZXMAMOZUNW
|
6.2 | IC50 | 3 | — | |
HIQKYBKHPZKDSE
|
6.2 | IC50 | 2 | — |