Target Details
| UniProt AC | P55210 |
|---|---|
| Gene Symbol | CASP7 |
| Protein Name | Caspase-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 306
- Clinical molecules 0
- Avg pChEMBL 7.38
KEGG Pathways (14)
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Legionellosis
- Lipid and atherosclerosis
- Non-alcoholic fatty liver disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Salmonella infection
- TNF signaling pathway
Active Molecules (306)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NVEIBIBNNZZXLH
|
7.4 | IC50 | 2 | — | |
UMHSZDAKIVGDNR
|
7.3 | Ki | 3 | — | |
KYJSQQPQAAKFQY
|
7.3 | IC50 | 2 | — | |
GIUGBCHQBCYCTJ
|
7.3 | IC50 | 2 | — | |
RRBOQMCBPIXZCY
|
7.3 | IC50 | 2 | — | |
BVPRPKGQOIQLMI
|
7.3 | IC50 | 2 | — | |
WJGNHRNPMJTWAO
|
7.3 | IC50 | 2 | — | |
TXWGTLBORQHCEB
|
7.3 | IC50 | 2 | — | |
AEYFPXLRNOQPNR
|
7.2 | IC50 | 2 | — | |
FXRYYTKWISSZGE
|
7.2 | IC50 | 2 | — | |
IRZYVIBRQPMBSG
|
7.2 | IC50 | 2 | — | |
YDTJDBMJRVDMKU
|
7.2 | IC50 | 2 | — | |
UMBVAPCONCILTL
|
7.2 | IC50 | 5 | — | |
LNQOGDMGNCKCJV
|
7.2 | IC50 | 2 | — | |
HERMWEDKDQDOTD
|
7.2 | IC50 | 2 | — | |
RBQBJJBLAZNQJZ
|
7.2 | IC50 | 2 | — | |
LWBNNPKCSRJWRE
|
7.2 | IC50 | 2 | — | |
NKBDSMREMMRFSI
|
7.2 | IC50 | 5 | — | |
NKBDSMREMMRFSI
|
7.2 | IC50 | 5 | — | |
STDJONDOUCKJSO
|
7.2 | IC50 | 3 | — | |
STDJONDOUCKJSO
|
7.2 | IC50 | 3 | — | |
LRIRHRYRLCJRQA
|
7.2 | IC50 | 2 | — | |
OZAFISSWLZQMIS
|
7.2 | IC50 | 5 | — | |
UUEMWRIOZLIPHU
|
7.2 | IC50 | 4 | — | |
UUEMWRIOZLIPHU
|
7.2 | IC50 | 4 | — | |
BEUDVJBODYYMBI
|
7.2 | IC50 | 2 | — | |
QXPRIMHKXWCGCU
|
7.2 | IC50 | 2 | — | |
LQXYDGHSLQNYCW
|
7.2 | IC50 | 2 | — | |
OEZQRTUGLYPVGI
|
7.2 | IC50 | 2 | — | |
DFEUSDFPTOGJKU
|
7.1 | IC50 | 2 | — | |
GWEMAMOVSFKYPL
|
7.1 | IC50 | 2 | — | |
NTFDHIOBCNIACN
|
7.1 | IC50 | 2 | — | |
YZQKWJFJWRAGSA
|
7.1 | IC50 | 2 | — | |
MIQOWTZVMDSHBY
|
7.1 | IC50 | 2 | — | |
WTXXKEPFHMWDDX
|
7.1 | IC50 | 2 | — | |
SAUQPQCMYXHHJG
|
7.1 | IC50 | 2 | — | |
AYQUXMOMSNPZEF
|
7.0 | Ki | 4 | — | |
NAJZBQCCBCKDIT
|
7.0 | Ki | 3 | — | |
URMGPEOQLIISAB
|
7.0 | Ki | 4 | — | |
VCWYKJKQZUPTQP
|
7.0 | Ki | 2 | — | |
YNRQFMSSDVQNGQ
|
7.0 | IC50 | 5 | — | |
NKBSCZIQSOVWKJ
|
7.0 | IC50 | 3 | — | |
NKBSCZIQSOVWKJ
|
7.0 | IC50 | 3 | — | |
CLVRDSQHWNEIQR
|
7.0 | IC50 | 2 | — | |
HLQVEUCDTUXVLS
|
7.0 | IC50 | 2 | — | |
PFAYCUAUBOGVDX
|
7.0 | IC50 | 2 | — | |
COLCPJSXGNKCEG
|
7.0 | IC50 | 2 | — | |
GTXNLQVCIHMROL
|
7.0 | IC50 | 2 | — | |
APKUVGMUIXJJAR
|
7.0 | IC50 | 2 | — | |
GQXBVBOSGIYTNU
|
7.0 | IC50 | 2 | — |