Target Details
| UniProt AC | P55210 |
|---|---|
| Gene Symbol | CASP7 |
| Protein Name | Caspase-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00656 (Peptidase_C14) |
Summary
- Multi-target molecules 306
- Clinical molecules 0
- Avg pChEMBL 7.38
KEGG Pathways (14)
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Cytosolic DNA-sensing pathway
- Efferocytosis
- Legionellosis
- Lipid and atherosclerosis
- Non-alcoholic fatty liver disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Salmonella infection
- TNF signaling pathway
Active Molecules (306)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XIMITGPWYYFUQF
|
10.9 | IC50 | 8 | — | |
YNRQFMSSDVQNGQ
|
10.1 | IC50 | 8 | — | |
NHHJXCJHJPGPEF
|
9.6 | IC50 | 4 | — | |
XWTJWAAMOCNKHH
|
9.5 | IC50 | 4 | — | |
OJYJCHGYJSCGSY
|
9.2 | IC50 | 2 | — | |
OEZQRTUGLYPVGI
|
9.0 | IC50 | 2 | — | |
INTJRTIYLCEHRJ
|
9.0 | IC50 | 4 | — | |
LVXZMAMJNHAXKU
|
9.0 | IC50 | 4 | — | |
CKRCPAGGKUFVIT
|
8.9 | IC50 | 4 | — | |
SFDIMTVHWVLTIP
|
8.9 | IC50 | 4 | — | |
MBFCFVOWKKZRNA
|
8.7 | IC50 | 2 | — | |
AEVFCJHPCHDXDJ
|
8.7 | IC50 | 2 | — | |
QAFBFHNIUINEJN
|
8.7 | IC50 | 4 | — | |
SCZQZYJOIBQIGS
|
8.6 | IC50 | 4 | — | |
ULPLTJMGFAFYSR
|
8.6 | IC50 | 2 | — | |
GEZSSSVQIGDDMR
|
8.6 | IC50 | 4 | — | |
KSIBLECLZAACGQ
|
8.6 | IC50 | 3 | — | |
MDRQEFUKIMUQFX
|
8.6 | IC50 | 4 | — | |
MTGSTDMYYFQKEE
|
8.6 | IC50 | 3 | — | |
UCOGGEXRPKAPHO
|
8.5 | IC50 | 3 | — | |
MPIKODMIUDLWKY
|
8.5 | IC50 | 3 | — | |
BTAFTKGHXXQLHC
|
8.5 | IC50 | 4 | — | |
SDEQMNUREZLDJE
|
8.5 | IC50 | 2 | — | |
GGRODTCKLDDOBP
|
8.5 | IC50 | 3 | — | |
JYGKCHPWCXRSQJ
|
8.4 | IC50 | 4 | — | |
XUUQUFQWQGVYPU
|
8.4 | IC50 | 2 | — | |
CBWLTWDVCXFXAG
|
8.4 | IC50 | 2 | — | |
CSEDBYKWGJUWMQ
|
8.4 | IC50 | 3 | — | |
HDXDXAKYCMKPSF
|
8.4 | IC50 | 4 | — | |
NJAQASWTRGUAGC
|
8.4 | IC50 | 3 | — | |
GQDJBEWJIKPEQS
|
8.3 | IC50 | 3 | — | |
NAZSWKZWCFVHEL
|
8.3 | IC50 | 4 | — | |
DPMMEOUVESBMSC
|
8.3 | IC50 | 2 | — | |
QLHDEYZCVHOGEF
|
8.3 | IC50 | 4 | — | |
JQQCMQLLJHRXIA
|
8.3 | IC50 | 2 | — | |
LHHQIZSDNGIYTJ
|
8.2 | IC50 | 2 | — | |
QGTNZCUWEMSWQW
|
8.2 | IC50 | 2 | — | |
ZUPAARUJOOKFLI
|
8.2 | IC50 | 2 | — | |
NORINPJAWOULPP
|
8.2 | IC50 | 2 | — | |
LYBWGROBJJXCJJ
|
8.2 | IC50 | 6 | — | |
IXNAXPALFGYLBG
|
8.1 | IC50 | 2 | — | |
AJJFEZDYZOETDJ
|
8.1 | IC50 | 2 | — | |
DPNDRYUDIJORHR
|
8.1 | IC50 | 2 | — | |
OOGHGBCRVSBUHH
|
8.1 | Ki | 3 | — | |
PSEYKDQFSOGYNR
|
8.1 | IC50 | 4 | — | |
BRCVHXRLGOWCTD
|
8.1 | IC50 | 2 | — | |
OMCJYUDICKFVIV
|
8.1 | IC50 | 2 | — | |
XRLQEVLRBDPXIT
|
8.1 | IC50 | 2 | — | |
VRYGMTNRJQGMBD
|
8.0 | IC50 | 2 | — | |
DKRXATGOSDBMOO
|
8.0 | IC50 | 2 | — |