Target Details
| UniProt AC | P55201 |
|---|---|
| Gene Symbol | BRPF1 |
| Protein Name | Peregrin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF10513 (EPL1) PF13831 (PHD_2) PF00855 (PWWP) PF13832 (zf-HC5HC2H_2) |
Summary
- Multi-target molecules 44
- Clinical molecules 0
- Avg pChEMBL 6.94
Associated Diseases (1)
Active Molecules (44)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QFOYNDFIBXQVIO
|
8.1 | IC50 | 3 | — | |
BINBUXZIKUNKAE
|
7.9 | IC50 | 2 | — | |
LQDXWIYREJVTTB
|
7.9 | IC50 | 4 | — | |
HYQBRUSSCIAOOD
|
7.8 | Kd | 6 | — | |
XULQOMADHZABKB
|
7.8 | IC50 | 3 | — | |
YPOOJPDFTKZDEW
|
7.8 | IC50 | 3 | — | |
WUCKMZXHDIJUHE
|
7.6 | IC50 | 2 | — | |
FFVNHKQONMKRRU
|
7.5 | IC50 | 2 | — | |
UEMQPCYDWCSVCU
|
7.5 | IC50 | 5 | — | |
BMVCSXFOQPYKKC
|
7.4 | IC50 | 5 | — | |
VXXXPCKZPJGNGK
|
7.4 | IC50 | 4 | — | |
GPMNHYJTFYQIDD
|
7.4 | IC50 | 2 | — | |
QCIJLRJBZDBVDB
|
7.3 | IC50 | 5 | — | |
NCCGOWLXEQZIMX
|
7.3 | IC50 | 2 | — | |
COVNONZQYCHIJS
|
7.2 | IC50 | 2 | — | |
OHKRNOLZIOHQBM
|
7.2 | IC50 | 2 | — | |
HHQVWOAKOPBQDP
|
7.2 | IC50 | 2 | — | |
MREZOHBMPINXNX
|
7.2 | IC50 | 2 | — | |
HVHLFMDXTXHXRM
|
7.2 | Kd | 2 | — | |
BXGJNRVCUDKEGW
|
7.0 | IC50 | 2 | — | |
KPWWFNXRLAAREN
|
7.0 | Kd | 12 | — | |
RBUYFHLQNPJMQM
|
7.0 | Kd | 10 | — | |
UYBRROMMFMPJAN
|
6.8 | IC50 | 8 | — | |
VZAFGXCWAWRULT
|
6.8 | Ki | 7 | — | |
AXJXDWNCHLEVAZ
|
6.8 | Kd | 4 | — | |
XWUSNMULJMQCCC
|
6.7 | IC50 | 3 | — | |
COGXRBWRVXDPDM
|
6.7 | IC50 | 2 | — | |
KNVIUMWNYXDULF
|
6.7 | IC50 | 2 | — | |
LVDUGYSBGLMRET
|
6.6 | Kd | 2 | — | |
HONYBLSJNSYWKQ
|
6.6 | Ki | 3 | — | |
YUNQZQREIHWDQT
|
6.6 | IC50 | 2 | — | |
GOSJWGMIGYNNGJ
|
6.5 | IC50 | 2 | — | |
MEWCCJKZDZAUIP
|
6.5 | IC50 | 2 | — | |
LMLIBNUOIWAJFC
|
6.4 | Kd | 9 | — | |
WMKFJDQPAVKQAQ
|
6.3 | IC50 | 3 | — | |
FSMTUHGXWGJNKK
|
6.2 | IC50 | 4 | — | |
UQJAUEXASXFSKA
|
6.2 | IC50 | 2 | — | |
YDDKRKCQSIKAJD
|
6.2 | IC50 | 3 | — | |
NZCCNFWSBAAKSI
|
6.2 | IC50 | 3 | — | |
KQJPZLNOKCNFSE
|
6.2 | IC50 | 2 | — | |
OKEWIHVRDQJMQG
|
6.2 | IC50 | 2 | — | |
JJGHZALDUUMGCU
|
6.1 | IC50 | 3 | — | |
SUIWTHQZBYYCGP
|
6.1 | Kd | 3 | — | |
OFZUZFZNFMUNAS
|
6.0 | IC50 | 3 | — |