Target Details
| UniProt AC | P55055 |
|---|---|
| Gene Symbol | NR1H2 |
| Protein Name | Oxysterols receptor LXR-beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 509
- Clinical molecules 0
- Avg pChEMBL 7.43
KEGG Pathways (2)
Active Molecules (509)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LBPQARCLPTVEGQ
|
6.7 | IC50 | 2 | — | |
ZJPIFOVRFHBVNC
|
6.7 | IC50 | 2 | — | |
DHBIWVAWNUNKJG
|
6.7 | IC50 | 2 | — | |
PNGBFYGVOOVAIY
|
6.7 | IC50 | 2 | — | |
QBUILYGRQMFSAV
|
6.7 | IC50 | 2 | — | |
AWFKUZKMHLKRBA
|
6.7 | IC50 | 2 | — | |
WJPMVXGXXLNBEN
|
6.7 | IC50 | 2 | — | |
DCFHWWUSMITHJJ
|
6.7 | IC50 | 2 | — | |
WZXCTCJIJVBAOX
|
6.7 | IC50 | 2 | — | |
LAHPLBHKJGGIEF
|
6.7 | IC50 | 2 | — | |
DUSQUBZCYLLKHT
|
6.6 | IC50 | 2 | — | |
ZLCICKWEGSYHOX
|
6.6 | IC50 | 2 | — | |
ZMLDZMJEIPYMEJ
|
6.6 | IC50 | 2 | — | |
YOYQINDKUAALSH
|
6.6 | Ki | 3 | — | |
JPIHSYRXQLKCID
|
6.6 | IC50 | 2 | — | |
MTPMZVFOMVXGMD
|
6.5 | IC50 | 2 | — | |
IEPOYBLCAUUPJP
|
6.5 | IC50 | 2 | — | |
RLNMZAJKGCKXRV
|
6.5 | IC50 | 2 | — | |
NKFDLBSCCAQKKW
|
6.5 | IC50 | 2 | — | |
GREUENDQALGMMV
|
6.5 | IC50 | 2 | — | |
GZAPSISRDWGGFB
|
6.5 | IC50 | 5 | — | |
SNVDXERLZQEYID
|
6.5 | IC50 | 2 | — | |
CQTCWVWUQDCTSG
|
6.5 | IC50 | 3 | — | |
GRHBEGZXUDYQLG
|
6.4 | IC50 | 2 | — | |
JVNKOHAYLUAZLM
|
6.4 | Ki | 2 | — | |
KCTVTEAWWHOHNZ
|
6.4 | IC50 | 2 | — | |
GMKDRYOJWQXLTE
|
6.4 | IC50 | 2 | — | |
FCQLLWXAPLXYQV
|
6.4 | IC50 | 2 | — | |
FFEMTQPBRTULCE
|
6.4 | IC50 | 2 | — | |
FLQMNHODIBPHAJ
|
6.4 | IC50 | 2 | — | |
PDAASAKPBNZZQB
|
6.3 | IC50 | 2 | — | |
XDSUZROBCUROQA
|
6.3 | IC50 | 2 | — | |
DNNYNSPBJXNYMZ
|
6.3 | IC50 | 2 | — | |
RZPAXNJLEKLXNO
|
6.3 | Ki | 2 | — | |
YJTSPUKQCBSIGP
|
6.3 | IC50 | 2 | — | |
YOBSSBAJFVWQAA
|
6.3 | IC50 | 2 | — | |
DYTISOKVYHWYCW
|
6.3 | IC50 | 2 | — | |
XBWKFFVZKTYRJE
|
6.2 | IC50 | 2 | — | |
AJPPENWWEOYGLC
|
6.2 | IC50 | 2 | — | |
BRUGTPFLMNPXDZ
|
6.2 | IC50 | 2 | — | |
BSOHTIRAIBGWNI
|
6.2 | IC50 | 2 | — | |
COAOXNQSRNFNRV
|
6.2 | IC50 | 2 | — | |
CYJDPJOAWCSPNC
|
6.2 | IC50 | 2 | — | |
FFVUWWDAZAEMFG
|
6.2 | IC50 | 2 | — | |
FKVVKQNEEGIOHR
|
6.2 | IC50 | 2 | — | |
FSXSVMWOIJNOPA
|
6.2 | IC50 | 2 | — | |
GFYAONIZMGHILK
|
6.2 | IC50 | 2 | — | |
GGYAYXDZATWEIK
|
6.2 | IC50 | 2 | — | |
GUZVQJUTIWTUCT
|
6.2 | IC50 | 2 | — | |
HUMBUMHTRIKMPI
|
6.2 | IC50 | 2 | — |