Target Details
| UniProt AC | P55055 |
|---|---|
| Gene Symbol | NR1H2 |
| Protein Name | Oxysterols receptor LXR-beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 509
- Clinical molecules 0
- Avg pChEMBL 7.43
KEGG Pathways (2)
Active Molecules (509)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TZRCVICHXMBFCB
|
6.9 | IC50 | 2 | — | |
MVQGOFQHJVGQCO
|
6.9 | IC50 | 2 | — | |
DGPCIFPFGHXRIB
|
6.9 | IC50 | 2 | — | |
MVZUVIXDADTQPL
|
6.9 | Ki | 2 | — | |
RFGMOPNIYZVCFS
|
6.9 | IC50 | 2 | — | |
UCPCLSOVORSWOU
|
6.9 | IC50 | 2 | — | |
PICJKSLPJSZRIV
|
6.9 | Ki | 2 | — | |
AETOIGDOKBMGSM
|
6.9 | IC50 | 2 | — | |
BFQFGSRUGHCILX
|
6.9 | IC50 | 2 | — | |
BZNZTFPVHCRTIJ
|
6.9 | IC50 | 2 | — | |
DLIGEYTVUWDKGR
|
6.9 | IC50 | 2 | — | |
DSAIHBOVBTWQFB
|
6.9 | IC50 | 2 | — | |
JKPRVFVLDDBCSV
|
6.9 | IC50 | 2 | — | |
KSMGMDVHOFLAFH
|
6.9 | IC50 | 2 | — | |
LWFAXHWAXCYXSZ
|
6.9 | Ki | 2 | — | |
NBZQZSXHBHHYKZ
|
6.9 | IC50 | 2 | — | |
NIOWYZWIYTYWKD
|
6.9 | IC50 | 2 | — | |
NTADGJLCICPJEW
|
6.9 | IC50 | 2 | — | |
OGIATJNVLIWGCR
|
6.9 | IC50 | 2 | — | |
PKIRPTWVIDGVIA
|
6.9 | IC50 | 2 | — | |
QRCKSIDYJUQFBB
|
6.9 | IC50 | 2 | — | |
SDRAOTAIGRLMCD
|
6.9 | IC50 | 2 | — | |
SRDMAHSGPGXUOC
|
6.9 | IC50 | 2 | — | |
SRIRHESFIMVQGY
|
6.9 | IC50 | 2 | — | |
UJPXVPZVYQWTNV
|
6.9 | IC50 | 2 | — | |
XCIASCLPGRSRQB
|
6.9 | IC50 | 2 | — | |
XPLRJSGSDRXZOR
|
6.9 | IC50 | 2 | — | |
YLHMEFUTYZUWEM
|
6.9 | IC50 | 2 | — | |
YUVUADPRHHCDCU
|
6.9 | IC50 | 2 | — | |
ZZDJDMMSFPXVHM
|
6.9 | IC50 | 2 | — | |
IKEBXOQTSPUHRL
|
6.9 | IC50 | 2 | — | |
PXRKUDZYCJZQBB
|
6.9 | IC50 | 2 | — | |
PZJQTRGWISHVPT
|
6.9 | IC50 | 2 | — | |
YYFFXRNVMLUSIQ
|
6.9 | Ki | 2 | — | |
SAKQPFIBVKAZMM
|
6.9 | Ki | 2 | — | |
JYNPEZDAIHSJHW
|
6.9 | IC50 | 2 | — | |
QQDXQGDFJZPVRX
|
6.9 | IC50 | 2 | — | |
WPUHRYSDQSXTGR
|
6.9 | IC50 | 2 | — | |
DWVNDOKJFPRSRU
|
6.8 | Ki | 2 | — | |
ZVLHOXBSTALIAV
|
6.8 | IC50 | 2 | — | |
CHCCPPPOKAASRP
|
6.8 | IC50 | 2 | — | |
LYILZTQKEIMJDW
|
6.8 | Ki | 3 | — | |
QDOPVBPHOQDBJS
|
6.8 | IC50 | 2 | — | |
GADXIGHAARSCIO
|
6.8 | IC50 | 3 | — | |
LUJCWOPVYNTRBQ
|
6.8 | Ki | 2 | — | |
XRYDEEKHRNPJOZ
|
6.8 | Ki | 3 | — | |
YYIDRXGXLIOEDJ
|
6.8 | IC50 | 2 | — | |
WWWVODUMLXMIRV
|
6.8 | Ki | 2 | — | |
AEORYXMWRGDQDS
|
6.8 | IC50 | 2 | — | |
YZWZMPWHXSZLBQ
|
6.8 | Ki | 3 | — |