Target Details
UniProt ACP55055
Gene SymbolNR1H2
Protein NameOxysterols receptor LXR-beta
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00104 (Hormone_recep) PF00105 (zf-C4)
Summary
  • Multi-target molecules 509
  • Clinical molecules 0
  • Avg pChEMBL 7.43
KEGG Pathways (2)
Top Co-occurrence Targets
Active Molecules (509)
InChIKey pChEMBL Type Targets Clinical
IDKRBDPKBAQNEZ 8.2 IC50 2
KMTFPMRUPSWRTQ 8.2 Ki 3
LWXOLPDIDYBJQJ 8.2 Ki 2
LYVSLMPYMYETMJ 8.2 Ki 3
NSWRBHFZGBXSGU 8.2 Ki 2
OEALQQJYLLGJFL 8.2 Ki 2
OMMCNHJJHLQJHQ 8.2 Ki 2
SENBJMMSGVHUDH 8.2 IC50 2
WZQNVHXAZPMTQI 8.2 Ki 2
DUOZJJLSLMAQCI 8.1 IC50 2
BGDPLINROWYUAR 8.1 Ki 2
HXOUVMGQDQYWNM 8.1 Ki 2
MMFGEAJCSXYUPB 8.1 Ki 2
MQKQOJAXHYOTRU 8.1 Ki 2
NLQZHFCXLSURKR 8.1 Ki 2
OVYOPGSHTATUOV 8.1 Ki 2
RKMWUDYBRYAWCA 8.1 Ki 2
WNHGOWAKQUWTHZ 8.1 Ki 2
YYDPUXBLDMRZQE 8.1 IC50 2
RPEJMRBNVYJBHP 8.1 Ki 2
YRWXCMJJJAVQPM 8.1 IC50 2
AJAGFKNPKFWBMC 8.1 IC50 2
JLWYCHMJOLWTSZ 8.1 IC50 2
CBDKGOMYQLDSHF 8.1 IC50 2
CRRQUBDXEDTMJH 8.1 Ki 2
GIPBQDFCFPOLCY 8.1 Ki 2
JSVXZVWRZPKCFT 8.1 Ki 2
QJGPMJDHZAMQSJ 8.1 Ki 2
QQRBREMSESSVRO 8.1 Ki 2
SKGJRIXOTUPIFB 8.1 Ki 2
SWBBNSPWRVCYAE 8.1 Ki 3
WZMZHHPXANSLBG 8.1 Ki 3
YIRPKYOIUDNERT 8.1 Ki 2
COULHFBFGNXFAF 8.0 Ki 2
JRJIJEXVKDFRTL 8.0 IC50 2
KKPXMFGSPSGBQW 8.0 IC50 2
KQGULCLQMZRZGO 8.0 Ki 2
OCSBWUNDZQJSRW 8.0 Ki 2
OHDRXCKGYPYQAU 8.0 IC50 2
UAHUOJIWTDTEMT 8.0 IC50 2
ULLMSRMSGPWBDE 8.0 Ki 2
WUVSLEJBHNUDBB 8.0 Ki 3
XSNDTQOGMFODQY 8.0 IC50 2
YPXOOPFXOOABHI 8.0 IC50 2
ZWGZCSXCYWYFTL 8.0 Ki 2
ZXTOKWKHXXGVMT 8.0 Ki 3
WAZXSGZGKNWHSO 8.0 Ki 2
BHKSYENPDNOBLX 8.0 IC50 2
CKHYMMLNOQQEMV 8.0 IC50 2
GEXZSCVAMWWQAV 8.0 Ki 2
2D structure