Target Details
UniProt ACP55055
Gene SymbolNR1H2
Protein NameOxysterols receptor LXR-beta
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00104 (Hormone_recep) PF00105 (zf-C4)
Summary
  • Multi-target molecules 509
  • Clinical molecules 0
  • Avg pChEMBL 7.43
KEGG Pathways (2)
Top Co-occurrence Targets
Active Molecules (509)
InChIKey pChEMBL Type Targets Clinical
GCAJNTSVNKDATQ 8.4 IC50 2
GCGBTTGCZAXGLQ 8.4 Ki 2
KZCSVWPMPDGZGU 8.4 Ki 2
MOQUFKNADUILIJ 8.4 IC50 2
NEGSIYPKPKVQAA 8.4 Ki 2
NVCNWULYEHGNKG 8.4 IC50 2
VSLBVBOGQLFVOY 8.4 Ki 2
XRWDAQASJVEARP 8.4 Ki 2
XVRHEEOCNTZUNF 8.4 Ki 2
ISMQLWMZRUKHEF 8.4 IC50 2
OEDBWXLEGYGITE 8.4 IC50 2
KIITVWQUUAGGON 8.4 IC50 2
LJZFYKYOXOCPDD 8.3 IC50 2
XZYFDTYSBRYCCK 8.3 IC50 2
UWFHFVAFWATDDO 8.3 IC50 2
BYZAOZSASXJAQT 8.3 IC50 2
CDLANIGSVPOVRJ 8.3 Ki 2
CQEKMSRTDPXHST 8.3 IC50 2
FMNHPFYLVZKAJK 8.3 IC50 2
FVKYONNSLLCHIF 8.3 IC50 2
LCDRBOYRRKJMEX 8.3 IC50 2
LIKCFBAAJFMUJP 8.3 IC50 2
VVVMBZVHNIYCQS 8.3 Ki 3
XOPXTKOQXWMGEF 8.3 Ki 2
YAKODSHNCZYDPB 8.3 IC50 2
YXXFEOBGLYBWLG 8.3 Ki 2
ZFAZSJUOGZNAMM 8.3 Ki 2
SELLUNCDLWGEEU 8.3 IC50 2
JVIDKHNOLQEIJP 8.3 IC50 2
IUMMDSSCERZSTJ 8.3 Ki 2
JNGMQNSQSCYLSD 8.3 IC50 2
AJSJAQQMFKYODQ 8.3 IC50 2
IQRSIUBKAADOQA 8.3 Ki 2
JQOXVKXWQCMPRP 8.2 IC50 2
AORBCLGGYNFMGN 8.2 IC50 4
HFGCUOYYZKNQLX 8.2 Ki 3
JUYXKAZFVVUFNZ 8.2 Ki 2
LNVWYDLYTZAVJQ 8.2 Ki 2
LODWYHGIAQYCAL 8.2 Ki 3
MWSOCMMZIFOCRI 8.2 Ki 2
NCZXBZJVJRJUSC 8.2 Ki 3
PAXOTBRHGNYSDC 8.2 Ki 2
PWFODDIPAXPLMJ 8.2 IC50 2
RPEJMRBNVYJBHP 8.2 Ki 2
TUYZXSLKXBNYSH 8.2 IC50 2
YXXFEOBGLYBWLG 8.2 Ki 2
ZIMHQMXADUASSG 8.2 IC50 2
HXANPPNXWQVOEO 8.2 IC50 2
CDVXSTXXLZGAKK 8.2 Ki 2
CCZANINLKOMNJX 8.2 Ki 2
2D structure