Target Details
| UniProt AC | P55055 |
|---|---|
| Gene Symbol | NR1H2 |
| Protein Name | Oxysterols receptor LXR-beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 509
- Clinical molecules 0
- Avg pChEMBL 7.43
KEGG Pathways (2)
Active Molecules (509)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NLDOCDWHNYIGKV
|
9.1 | IC50 | 2 | — | |
ASTLYMNMTDERKI
|
9.0 | IC50 | 2 | — | |
CXSWMXMKWWOTPK
|
9.0 | IC50 | 2 | — | |
MVEYCHUAHRZQOD
|
9.0 | Ki | 3 | — | |
SWVQEDYQXWDKTA
|
9.0 | Ki | 2 | — | |
VTSLTFRMYLXJLX
|
9.0 | Ki | 2 | — | |
XOTHLYNSDMSVGX
|
9.0 | Ki | 2 | — | |
YTEDTWJJQBCOTI
|
9.0 | Ki | 2 | — | |
JQOOZVXMCPGTNO
|
8.8 | IC50 | 2 | — | |
MFLGRDLZNMSORM
|
8.8 | IC50 | 2 | — | |
MYNWRKZLIIDPBU
|
8.8 | IC50 | 2 | — | |
BKINFWHEJAZZTL
|
8.8 | IC50 | 2 | — | |
NVDRYPHMVKODMP
|
8.7 | IC50 | 2 | — | |
AVHJCISEWCJAIL
|
8.7 | IC50 | 2 | — | |
USWOEXHVBVCJOR
|
8.7 | IC50 | 2 | — | |
DZOUMAUJJDVJHY
|
8.7 | IC50 | 2 | — | |
LFYZXWABUGTSOT
|
8.7 | IC50 | 2 | — | |
NXAQUWGSGCUYGJ
|
8.7 | Ki | 2 | — | |
OUJQRQRBNRGQTC
|
8.7 | IC50 | 2 | — | |
OWWNUAVAXAAAAM
|
8.7 | IC50 | 2 | — | |
SBYNVOVSJLOHRE
|
8.7 | IC50 | 2 | — | |
UUIQBDLORYXQJP
|
8.7 | IC50 | 2 | — | |
XTWZRTUIFQOMNH
|
8.7 | Ki | 2 | — | |
VXHRQVMQVYQGQG
|
8.7 | IC50 | 2 | — | |
DHCPTZAZDOXILJ
|
8.7 | IC50 | 2 | — | |
DRNWBBRZORIYEI
|
8.6 | IC50 | 2 | — | |
QMAWFUWIOSWDJM
|
8.6 | IC50 | 2 | — | |
ZDUOYBOFMKORCT
|
8.6 | IC50 | 2 | — | |
MMQLCGFOEBSWCN
|
8.6 | IC50 | 2 | — | |
MFDLTITVUNIPCT
|
8.6 | IC50 | 2 | — | |
QIFYDQQBXMOQLW
|
8.6 | IC50 | 2 | — | |
QQNXCYFWSCPJOI
|
8.6 | IC50 | 2 | — | |
SQHRBEDYCPJCNA
|
8.6 | IC50 | 2 | — | |
DIEQFJUHAMDHJZ
|
8.6 | IC50 | 2 | — | |
GEDMLXRPUQZAAS
|
8.6 | IC50 | 2 | — | |
DDVQRICMCZPTNJ
|
8.5 | IC50 | 2 | — | |
AAXKPQBGHZNCOJ
|
8.5 | IC50 | 2 | — | |
GVRPVYDNQAVCMD
|
8.5 | Ki | 2 | — | |
IGGSXCWSHVYVMA
|
8.5 | Ki | 2 | — | |
ITROVDJOIPDCOB
|
8.5 | IC50 | 2 | — | |
VCNKBGCNOUBXAD
|
8.5 | Ki | 2 | — | |
APHRFSGOWKZUGE
|
8.5 | IC50 | 2 | — | |
GBEWPJJHRRWGJD
|
8.5 | IC50 | 2 | — | |
AIZFRFCHCJRXFS
|
8.5 | IC50 | 2 | — | |
GKRQECRQGLCHTJ
|
8.5 | IC50 | 2 | — | |
JWRIUHZELXTXLP
|
8.5 | IC50 | 2 | — | |
PBQUJALWEDBRLW
|
8.5 | IC50 | 2 | — | |
FWTLKBYOKWCAEO
|
8.4 | IC50 | 2 | — | |
CHDZBJMLJJYFFA
|
8.4 | IC50 | 2 | — | |
DPAWQSUVLANLRD
|
8.4 | IC50 | 2 | — |