Target Details
| UniProt AC | P54764 |
|---|---|
| Gene Symbol | EPHA4 |
| Protein Name | Ephrin type-A receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF07647 (SAM_2) |
Summary
- Multi-target molecules 33
- Clinical molecules 13
- Avg pChEMBL 7.01
KEGG Pathways (1)
Active Molecules (33)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBNZXTGUTAYRHI
|
8.9 | Kd | 102 | Yes | |
SEJGTFPOEJWEGG
|
8.7 | Kd | 149 | — | |
AQSSMEORRLJZLU
|
8.7 | Kd | 34 | Yes | |
JTWMOWRMSZZHDR
|
8.5 | IC50 | 13 | — | |
SFCBIFOAGRZJNX
|
8.3 | Kd | 22 | — | |
VAARYSWULJUGST
|
8.1 | Kd | 119 | Yes | |
BETBNWGUKZUUAX
|
8.1 | IC50 | 21 | — | |
UBPYILGKFZZVDX
|
7.7 | Kd | 130 | Yes | |
WKDACQVEJIVHMZ
|
7.7 | Kd | 46 | — | |
CXQHYVUVSFXTMY
|
7.4 | Kd | 154 | — | |
MVCOAUNKQVWQHZ
|
7.2 | IC50 | 54 | Yes | |
ZCCPLJOKGAACRT
|
7.1 | IC50 | 599 | — | |
MRTHXFZEQBERDI
|
7.1 | IC50 | 11 | — | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
XKFTZKGMDDZMJI
|
6.8 | Kd | 64 | Yes | |
ALKJNCZNEOTEMP
|
6.8 | Kd | 55 | — | |
DKZYXHCYPUVGAF
|
6.7 | Kd | 112 | — | |
YHVHYWYQEFELOW
|
6.6 | IC50 | 44 | — | |
HKSZLNNOFSGOKW
|
6.5 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.5 | Kd | 213 | — | |
OMZCMEYTWSXEPZ
|
6.5 | Kd | 43 | Yes | |
HHZIURLSWUIHRB
|
6.5 | Kd | 57 | Yes | |
KTEIFNKAUNYNJU
|
6.4 | Kd | 114 | — | |
ODPGGGTTYSGTGO
|
6.4 | Kd | 153 | — | |
HHFBDROWDBDFBR
|
6.4 | Kd | 40 | Yes | |
HVXKQKFEHMGHSL
|
6.4 | Kd | 21 | — | |
ZLHFILGSQDJULK
|
6.3 | Kd | 37 | Yes | |
OUKYUETWWIPKQR
|
6.0 | Kd | 31 | Yes | |
QQWUGDVOUVUTOY
|
6.0 | Kd | 231 | Yes | |
MFAQYJIYDMLAIM
|
6.0 | Kd | 130 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |