Target Details
| UniProt AC | P54762 |
|---|---|
| Gene Symbol | EPHB1 |
| Protein Name | Ephrin type-B receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 26
- Clinical molecules 12
- Avg pChEMBL 7.03
KEGG Pathways (1)
Active Molecules (26)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBNZXTGUTAYRHI
|
9.3 | Kd | 102 | Yes | |
JTWMOWRMSZZHDR
|
9.0 | IC50 | 13 | — | |
VAARYSWULJUGST
|
8.4 | Kd | 119 | Yes | |
RFSFIDGEFVXSQM
|
8.2 | IC50 | 12 | Yes | |
CXQHYVUVSFXTMY
|
7.9 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.9 | Kd | 149 | — | |
HHZIURLSWUIHRB
|
7.8 | Ki | 57 | Yes | |
UBPYILGKFZZVDX
|
7.5 | Kd | 130 | Yes | |
MIMOHMCANSGXIG
|
7.4 | IC50 | 15 | — | |
MVCOAUNKQVWQHZ
|
7.0 | IC50 | 54 | Yes | |
KTEIFNKAUNYNJU
|
6.9 | Kd | 114 | — | |
HKSZLNNOFSGOKW
|
6.9 | IC50 | 408 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
HKSZLNNOFSGOKW
|
6.6 | Kd | 213 | — | |
UHTHHESEBZOYNR
|
6.5 | Kd | 66 | Yes | |
HHFBDROWDBDFBR
|
6.5 | Kd | 40 | Yes | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
NHHQJBCNYHBUSI
|
6.4 | Kd | 220 | — | |
WPXVVAWAHQHJPF
|
6.4 | IC50 | 41 | — | |
WINHZLLDWRZWRT
|
6.3 | Kd | 201 | Yes | |
XZXHXSATPCNXJR
|
6.3 | Kd | 165 | Yes | |
VCZDFACOFNRTMG
|
6.2 | IC50 | 6 | — | |
MPVGZUGXCQEXTM
|
6.1 | Kd | 61 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |