Target Details
| UniProt AC | P54760 |
|---|---|
| Gene Symbol | EPHB4 |
| Protein Name | Ephrin type-B receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 533
- Clinical molecules 99
- Avg pChEMBL 6.88
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (533)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PQYBSOBFELGWEF
|
6.3 | IC50 | 2 | — | |
PRVHVZIMFXZSQV
|
6.3 | IC50 | 3 | — | |
PVTTWYOJLADNCZ
|
6.3 | IC50 | 4 | — | |
PWNBTHIQJMPMTI
|
6.3 | IC50 | 4 | — | |
QFHBQKXGJZQISJ
|
6.3 | IC50 | 3 | — | |
QHBIMTBQLBHDHJ
|
6.3 | IC50 | 2 | — | |
QHTZGTDGFHTCOG
|
6.3 | IC50 | 3 | — | |
QJMKYRIHQWAKSM
|
6.3 | IC50 | 3 | — | |
QMONPAAOIIDBIL
|
6.3 | IC50 | 3 | — | |
QOEMXTGSYTXSBD
|
6.3 | IC50 | 4 | — | |
QOLKGXDWVMWHLS
|
6.3 | IC50 | 3 | — | |
QPNYAXXXUXFKDG
|
6.3 | IC50 | 5 | — | |
QPQAGSRLQDSAGQ
|
6.3 | IC50 | 2 | — | |
QUDDVDXFQIWBKM
|
6.3 | IC50 | 2 | — | |
RFGYFZFUMBQSCW
|
6.3 | IC50 | 6 | — | |
RFKWUHOHGOAWTQ
|
6.3 | IC50 | 3 | — | |
RGUFKCMSOMSTHM
|
6.3 | IC50 | 3 | — | |
RJGUQSMXHFQXPD
|
6.3 | IC50 | 3 | — | |
RORFVUDLEIRGQY
|
6.3 | IC50 | 3 | — | |
RPLCLUCJTHAIOW
|
6.3 | IC50 | 3 | — | |
RSQKKUZJTBAHBG
|
6.3 | IC50 | 5 | — | |
RVMLSAUWFLLGAT
|
6.3 | IC50 | 5 | — | |
RZKGVOJSKFTTBA
|
6.3 | IC50 | 3 | — | |
SDPXNCYWHLAZJC
|
6.3 | IC50 | 4 | — | |
SHKAUSIXYOWPKS
|
6.3 | IC50 | 3 | — | |
SJEYKCLWHCAMQL
|
6.3 | IC50 | 3 | — | |
SLWMPPADXCAMND
|
6.3 | IC50 | 3 | — | |
SMLYFAJYRKAOPL
|
6.3 | IC50 | 2 | — | |
SPUVKXRMQZAIAZ
|
6.3 | IC50 | 4 | — | |
SYTDXYNETZANOI
|
6.3 | IC50 | 3 | — | |
TUJUURQEVYFCIN
|
6.3 | IC50 | 3 | — | |
TUQBWKPRXZNXMC
|
6.3 | IC50 | 2 | — | |
TZOPEIOUJFXKQZ
|
6.3 | IC50 | 3 | — | |
UHTHHESEBZOYNR
|
6.3 | Kd | 66 | Yes | |
UIELDVYKNRNSEM
|
6.3 | IC50 | 3 | — | |
UKKBXHWKVGSVEV
|
6.3 | IC50 | 4 | — | |
UQJWQNWEZPXTRQ
|
6.3 | IC50 | 3 | — | |
UUILILXZMGYNLD
|
6.3 | IC50 | 2 | — | |
VATKWVNDCITFEB
|
6.3 | IC50 | 3 | — | |
VEIQGMIXACRMMO
|
6.3 | IC50 | 5 | — | |
VEZBREXQDQRJTD
|
6.3 | IC50 | 2 | — | |
VOQVXZHQBTXEHV
|
6.3 | IC50 | 3 | — | |
VQRNHLREZMWHGF
|
6.3 | IC50 | 3 | — | |
VWCXCYRYWPKZNG
|
6.3 | IC50 | 3 | — | |
VXJCKEGWFQFYGD
|
6.3 | IC50 | 4 | — | |
VYVLFCZOKFCBJQ
|
6.3 | IC50 | 3 | — | |
WFNAULMUNPRODX
|
6.3 | IC50 | 2 | — | |
WQHZIFFISAIJEF
|
6.3 | IC50 | 4 | — | |
WUCSNTVXKXMTBP
|
6.3 | IC50 | 3 | — | |
WVCAYXOTVLLXMU
|
6.3 | IC50 | 4 | — |