Target Details
| UniProt AC | P54760 |
|---|---|
| Gene Symbol | EPHB4 |
| Protein Name | Ephrin type-B receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 533
- Clinical molecules 99
- Avg pChEMBL 6.88
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (533)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CWWBHDIXVWOCMI
|
6.4 | IC50 | 2 | — | |
IVPZQVJSLCFTTO
|
6.4 | IC50 | 10 | Yes | |
SPMVMDHWKHCIDT
|
6.4 | IC50 | 30 | — | |
CXUVPVMNMZKERT
|
6.4 | IC50 | 3 | Yes | |
NNQHKTWARZSGTQ
|
6.4 | IC50 | 7 | — | |
ZUMICAGHFTUJTI
|
6.4 | IC50 | 4 | Yes | |
FOMAIMPXVLHOCI
|
6.4 | IC50 | 10 | Yes | |
AAHKGRWRYBCWDL
|
6.3 | IC50 | 11 | Yes | |
UBJGLXSFXKIIFY
|
6.3 | IC50 | 12 | Yes | |
VOPNWXZDJKCCRE
|
6.3 | IC50 | 7 | Yes | |
FHNLPTRXVQOXQO
|
6.3 | IC50 | 11 | Yes | |
COAQRADEUYYCDG
|
6.3 | IC50 | 12 | Yes | |
ABXIBRWZRWHJCZ
|
6.3 | IC50 | 5 | — | |
AFHNMWQBLLGGSP
|
6.3 | IC50 | 5 | — | |
AHIOWTSQFILAEW
|
6.3 | IC50 | 5 | — | |
AVADFQHEIADTFF
|
6.3 | IC50 | 3 | — | |
AXFITPBCUMOSEI
|
6.3 | IC50 | 3 | — | |
BDVHNGIDDSJCCD
|
6.3 | IC50 | 3 | — | |
BKBIBLPFCFCOQQ
|
6.3 | IC50 | 3 | — | |
BLBVISQGOQQTND
|
6.3 | IC50 | 5 | — | |
BLZCIAZUKSOFTP
|
6.3 | IC50 | 2 | — | |
BQCYIIVLNTWNSU
|
6.3 | IC50 | 3 | — | |
BVPDJKPURONCRY
|
6.3 | IC50 | 4 | — | |
BYRDCUSCDUCHLA
|
6.3 | IC50 | 4 | — | |
CMTRUERFSJKMJQ
|
6.3 | IC50 | 5 | — | |
COWKEXRPFBNPOQ
|
6.3 | IC50 | 3 | — | |
DBXVNVVGMHBBOC
|
6.3 | IC50 | 3 | — | |
DICBCRYPBMEARO
|
6.3 | IC50 | 2 | — | |
DVEHRUCQBHJWFA
|
6.3 | IC50 | 5 | — | |
FAJVOBZBVGQKFD
|
6.3 | IC50 | 3 | — | |
FGHXOSBHGQKMBX
|
6.3 | IC50 | 4 | — | |
FJUIAQIBGJSIJS
|
6.3 | IC50 | 3 | — | |
FRHNEIRUMPIDKL
|
6.3 | IC50 | 3 | — | |
FSJDACURTSWGHC
|
6.3 | IC50 | 5 | — | |
FSJDACURTSWGHC
|
6.3 | IC50 | 4 | — | |
FSNXDZZUWFZSPA
|
6.3 | IC50 | 3 | — | |
FYJMEEVVSSJUMQ
|
6.3 | IC50 | 4 | — | |
FZGGLLMOLZVRHY
|
6.3 | IC50 | 3 | — | |
GBVHHGINCYVVRZ
|
6.3 | IC50 | 2 | — | |
GCBUMMPSFVNQKY
|
6.3 | IC50 | 2 | — | |
GKDGCIISLGIYBM
|
6.3 | IC50 | 3 | — | |
GNBFLDHHHUBBFG
|
6.3 | IC50 | 3 | — | |
HFTHZTJJBJKTGD
|
6.3 | IC50 | 3 | — | |
HJOMYFVOXGNASK
|
6.3 | IC50 | 2 | — | |
HLDHNATWCDWAML
|
6.3 | IC50 | 3 | — | |
HMNGFRURISAKFO
|
6.3 | IC50 | 3 | — | |
HQHKCYQAKIHFNI
|
6.3 | IC50 | 3 | — | |
HSVSYWHNTHEXTN
|
6.3 | IC50 | 3 | — | |
HTKJGEPLONIJLG
|
6.3 | IC50 | 3 | — | |
HVXKQKFEHMGHSL
|
6.3 | IC50 | 5 | — |