Target Details
| UniProt AC | P54760 |
|---|---|
| Gene Symbol | EPHB4 |
| Protein Name | Ephrin type-B receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 533
- Clinical molecules 99
- Avg pChEMBL 6.88
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (533)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DJCCECXADYTNDZ
|
7.0 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
7.0 | Kd | 154 | — | |
HHCBMISMPSAZBF
|
7.0 | IC50 | 23 | — | |
RHAMYMXUVZEEJR
|
7.0 | IC50 | 4 | — | |
RHGZQGXELRMGES
|
7.0 | IC50 | 8 | Yes | |
MRCFTWAYZAHAFA
|
7.0 | IC50 | 12 | Yes | |
DYMJWJDJSBQQRF
|
7.0 | IC50 | 2 | — | |
SXLHBXZCPKJTRT
|
7.0 | IC50 | 2 | — | |
ZBTLTVIYBHYEHL
|
7.0 | IC50 | 13 | Yes | |
UQRCJCNVNUFYDX
|
7.0 | Kd | 27 | — | |
YHHHJKZCRBUOTD
|
6.9 | IC50 | 2 | — | |
XZIADLYCTOCKRV
|
6.9 | IC50 | 5 | — | |
MIMOHMCANSGXIG
|
6.9 | IC50 | 15 | — | |
GHPCAIWYHJZRGR
|
6.9 | IC50 | 3 | Yes | |
PCSKFQHKWWNIKM
|
6.9 | IC50 | 7 | — | |
DKZYXHCYPUVGAF
|
6.8 | Kd | 112 | — | |
MRTHXFZEQBERDI
|
6.8 | IC50 | 11 | — | |
ISBXIYLTBRTLRK
|
6.8 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.8 | IC50 | 408 | — | |
CJMMCIXRPVLDBH
|
6.8 | IC50 | 12 | Yes | |
RHFWTFDTRBFIHU
|
6.8 | IC50 | 13 | Yes | |
DRWYYBMXZJLBHL
|
6.8 | IC50 | 3 | — | |
ZSAJPWOGVMFXHN
|
6.8 | IC50 | 10 | Yes | |
FLYHDJWABMRYPV
|
6.7 | IC50 | 2 | — | |
NVRXTLZYXZNATH
|
6.7 | IC50 | 47 | Yes | |
CKFCXTPUBPBSNV
|
6.7 | IC50 | 2 | — | |
ZLMVXCGWUJXFNP
|
6.7 | IC50 | 15 | Yes | |
PNEGWAQERPTPDN
|
6.6 | IC50 | 12 | Yes | |
GEZALMMCQYDFML
|
6.6 | IC50 | 15 | Yes | |
MNJNKKYCZKBVRY
|
6.6 | IC50 | 10 | Yes | |
BTIKYUUNPGWLNG
|
6.6 | IC50 | 12 | Yes | |
MJALZBJFTIQSSR
|
6.6 | IC50 | 12 | Yes | |
COAQRADEUYYCDG
|
6.6 | IC50 | 12 | Yes | |
FRKWMLCUONAHJH
|
6.6 | IC50 | 13 | Yes | |
XNODQMMIMXSTMX
|
6.6 | IC50 | 12 | Yes | |
ALKJNCZNEOTEMP
|
6.5 | Kd | 55 | — | |
GMVQPWCWWLPOQT
|
6.5 | IC50 | 9 | Yes | |
UVFCDQJUKYMBAZ
|
6.5 | IC50 | 10 | Yes | |
ZQQZSFIPDUAFMC
|
6.5 | IC50 | 3 | — | |
FAWGCSGOLCHXBH
|
6.5 | IC50 | 11 | Yes | |
MWYBBCLGEHZSCP
|
6.5 | IC50 | 11 | Yes | |
HRRMXIICSWVXIS
|
6.5 | IC50 | 13 | Yes | |
YQYKQJHEHMVZCD
|
6.5 | IC50 | 2 | — | |
KTTGLAHMSDMRLJ
|
6.5 | IC50 | 12 | Yes | |
LPFWVDIFUFFKJU
|
6.5 | Kd | 9 | — | |
ZPTUIPHHTLAHSJ
|
6.5 | IC50 | 3 | — | |
LVUGPVDXTSJQQD
|
6.5 | IC50 | 13 | Yes | |
QHIMVPIOWKYPSO
|
6.5 | IC50 | 2 | Yes | |
PFRDPPRTLFHGLR
|
6.5 | IC50 | 10 | Yes | |
YJNVZAXZUDOAAI
|
6.5 | IC50 | 10 | Yes |