Target Details
| UniProt AC | P54760 |
|---|---|
| Gene Symbol | EPHB4 |
| Protein Name | Ephrin type-B receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 533
- Clinical molecules 99
- Avg pChEMBL 6.88
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (533)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WPKITCNGCYKRNZ
|
7.3 | IC50 | 3 | — | |
WTOQAKRNPRFBML
|
7.3 | IC50 | 3 | — | |
WVXLPNDNCDLCQW
|
7.3 | IC50 | 2 | — | |
XCAOLOJNZVNRSK
|
7.3 | IC50 | 5 | — | |
XDESVXWYQFZXJJ
|
7.3 | IC50 | 4 | — | |
XJDLHHHTZRBRFC
|
7.3 | IC50 | 4 | — | |
XNWJPKXDERVJBQ
|
7.3 | IC50 | 3 | — | |
XRRHFQQSBXKXCI
|
7.3 | IC50 | 4 | — | |
XRTAZINADDFLOG
|
7.3 | IC50 | 3 | — | |
XYNKEFOTYHJQFS
|
7.3 | IC50 | 3 | — | |
YAEMBTULTQVMDI
|
7.3 | IC50 | 3 | — | |
YJHVTCUKZLXENT
|
7.3 | IC50 | 2 | — | |
YVZZAELYZKUMKK
|
7.3 | IC50 | 3 | — | |
ZEFUNPUAOZNDER
|
7.3 | IC50 | 4 | — | |
ZEFUNPUAOZNDER
|
7.3 | IC50 | 4 | — | |
ZFLUWPGMYIIBJD
|
7.3 | IC50 | 4 | — | |
ZJOIMYDGIVGAMA
|
7.3 | IC50 | 3 | — | |
ZKUNKJWGKBMFCR
|
7.3 | IC50 | 4 | — | |
ZPNITDGPLQDXIJ
|
7.3 | IC50 | 2 | — | |
ZPNSUJMOMIXELJ
|
7.3 | IC50 | 4 | — | |
ZWBURYJEEIVZFT
|
7.3 | IC50 | 4 | — | |
MBPKPSDAPFPECJ
|
7.3 | IC50 | 12 | Yes | |
UMBFDGUGXMOMHX
|
7.3 | IC50 | 12 | — | |
KCEWOOVCWCPFCY
|
7.2 | IC50 | 5 | — | |
NYEBJLYZEHKODB
|
7.2 | IC50 | 5 | Yes | |
FIWCLCRWDUELGO
|
7.2 | IC50 | 2 | — | |
NWEIPABWNQPRCZ
|
7.2 | IC50 | 7 | Yes | |
OTTCBLPTHPBEEX
|
7.2 | Ki | 11 | Yes | |
PQRFMBAACAPZPP
|
7.2 | IC50 | 12 | Yes | |
WVXNSAVVKYZVOE
|
7.2 | IC50 | 92 | — | |
YJSFAHMGDRBZGH
|
7.2 | IC50 | 16 | Yes | |
BOQLSYBMPFBUNE
|
7.2 | IC50 | 4 | — | |
VATOEUXNKZGEPM
|
7.2 | IC50 | 2 | — | |
NDUAHACMVSARNG
|
7.2 | IC50 | 4 | — | |
OSUPNTUMBGPMEA
|
7.1 | IC50 | 3 | — | |
OTJLQOSBMKGOAA
|
7.1 | IC50 | 2 | — | |
DYHVAHJSHIYCLL
|
7.1 | IC50 | 4 | — | |
BGDBURMJOLMENX
|
7.1 | IC50 | 3 | Yes | |
ZPXXVJYFXNATQZ
|
7.1 | IC50 | 3 | — | |
SMTDHTZNDOVANM
|
7.1 | IC50 | 2 | — | |
AIKGYQDFIJRQIY
|
7.1 | IC50 | 9 | — | |
NJRWVVJEQIMSFC
|
7.1 | IC50 | 2 | — | |
ZXTNBCJQGUOHPF
|
7.1 | IC50 | 2 | — | |
QTFCKBFCXDAZIU
|
7.0 | IC50 | 2 | — | |
RQXYLZHJULSWPX
|
7.0 | IC50 | 2 | — | |
ILWOIMOKLTUADE
|
7.0 | IC50 | 4 | — | |
OGKWTSFTGHKPIC
|
7.0 | IC50 | 3 | — | |
YBUFHSXYBABPHF
|
7.0 | IC50 | 3 | — | |
IWGLXKVBQSBQMC
|
7.0 | IC50 | 13 | Yes | |
JCMWWPAJCOQLAF
|
7.0 | IC50 | 11 | Yes |