Target Details
| UniProt AC | P54760 |
|---|---|
| Gene Symbol | EPHB4 |
| Protein Name | Ephrin type-B receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 533
- Clinical molecules 99
- Avg pChEMBL 6.88
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (533)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZCGKVBJAWNXBSX
|
7.8 | IC50 | 3 | — | |
UDUPSRWUDACGIS
|
7.8 | IC50 | 13 | Yes | |
XKFTZKGMDDZMJI
|
7.8 | Kd | 64 | Yes | |
ANJMTRKKSQNBTH
|
7.7 | IC50 | 3 | — | |
BNRXMSGHPVYSDK
|
7.6 | IC50 | 24 | — | |
QDQFGRCUJGQRLD
|
7.6 | IC50 | 3 | — | |
PAKQTWXBGSSCPQ
|
7.6 | IC50 | 2 | — | |
NDXRDWNCKIAIEH
|
7.6 | IC50 | 3 | — | |
IAVMNGJNMUJPOX
|
7.6 | IC50 | 3 | Yes | |
VREZKFPACUPTJS
|
7.5 | IC50 | 5 | — | |
UVHLKFVTSZBBCD
|
7.5 | IC50 | 2 | — | |
VZRIBSCWFNIDIU
|
7.5 | IC50 | 3 | — | |
WYLBYVHRCHPXRQ
|
7.5 | IC50 | 3 | — | |
RFSFIDGEFVXSQM
|
7.5 | IC50 | 12 | Yes | |
ZBRROTSBDAODQD
|
7.5 | IC50 | 7 | Yes | |
LWLYTBIEINCWJQ
|
7.5 | IC50 | 3 | Yes | |
OHZQTNDZRUYHEH
|
7.4 | IC50 | 3 | Yes | |
HVXKQKFEHMGHSL
|
7.4 | Kd | 21 | — | |
LIMHWCZODBAXBC
|
7.4 | IC50 | 3 | — | |
QTTGVGLTCILDCA
|
7.4 | IC50 | 7 | — | |
SPIWOLIEUWRHGI
|
7.4 | IC50 | 3 | Yes | |
YNGDGIGDNVCQGR
|
7.4 | IC50 | 3 | — | |
FICBCKOSWMLHMT
|
7.4 | IC50 | 3 | — | |
VDQZIQXNPVFCAD
|
7.4 | IC50 | 3 | Yes | |
ZHARSIGHGZRJLM
|
7.3 | IC50 | 2 | — | |
ZTQOHJNXDAUMOA
|
7.3 | IC50 | 13 | Yes | |
GTDRUFDOKAMNII
|
7.3 | IC50 | 3 | — | |
NCDVMWSJHOBWBM
|
7.3 | IC50 | 3 | — | |
UMGGFVAOWVEZEZ
|
7.3 | IC50 | 3 | — | |
AAWZYZGJDOSLSU
|
7.3 | IC50 | 4 | — | |
AKMSPGIAHZAWSW
|
7.3 | IC50 | 3 | — | |
ATNQJIZWZJGBST
|
7.3 | IC50 | 4 | — | |
AYWUHPUXKGVOSD
|
7.3 | IC50 | 3 | — | |
BACURHXRJBKWQO
|
7.3 | IC50 | 4 | — | |
BADQNHXUQWKUBJ
|
7.3 | IC50 | 3 | — | |
BFJHJPQKOHADCT
|
7.3 | IC50 | 3 | — | |
BLPHPXYTDDFZER
|
7.3 | IC50 | 2 | — | |
BTGGKWOJEKOLEQ
|
7.3 | IC50 | 3 | — | |
BZYUMECEYCQIQF
|
7.3 | IC50 | 3 | — | |
CJQXHWIFGRLKGH
|
7.3 | IC50 | 3 | — | |
CKIBKYNCWLLXRU
|
7.3 | IC50 | 3 | — | |
CKTFKRFHQMIOAN
|
7.3 | IC50 | 5 | — | |
CMTRUERFSJKMJQ
|
7.3 | IC50 | 4 | — | |
CPDVUYTVYREKJG
|
7.3 | IC50 | 3 | — | |
CXTBYZCZYIJFDG
|
7.3 | IC50 | 5 | — | |
DCHUHENWAKOFLF
|
7.3 | IC50 | 4 | — | |
DLZJESFGQYKOIJ
|
7.3 | IC50 | 3 | — | |
DNTJORWEWRMHBN
|
7.3 | IC50 | 4 | — | |
DUNQTRHEGUIEHU
|
7.3 | IC50 | 4 | — | |
FBKDSVZIPCLRHF
|
7.3 | IC50 | 3 | — |