Target Details
| UniProt AC | P54760 |
|---|---|
| Gene Symbol | EPHB4 |
| Protein Name | Ephrin type-B receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 533
- Clinical molecules 99
- Avg pChEMBL 6.88
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (533)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WYZCWZRHCBLLRQ
|
6.3 | IC50 | 3 | — | |
XHBINYIIFGVWSM
|
6.3 | IC50 | 5 | — | |
XJAYAHAZZKYCJC
|
6.3 | IC50 | 3 | — | |
XXVRAEWUOFARHO
|
6.3 | IC50 | 3 | — | |
YETQQFMHUDZVIA
|
6.3 | IC50 | 5 | — | |
YNRDGUQMVYIVCM
|
6.3 | IC50 | 3 | — | |
YXCHYSQVLDVUOJ
|
6.3 | IC50 | 3 | — | |
ZAMYFBONNUIDDG
|
6.3 | IC50 | 5 | — | |
ZDTMGSSRQLKYTK
|
6.3 | IC50 | 5 | — | |
ZLFBWBUGVAULCA
|
6.3 | IC50 | 2 | — | |
ZMGKRGOCDQRNTB
|
6.3 | IC50 | 3 | — | |
ZNKFCCNXFVRXHC
|
6.3 | IC50 | 3 | — | |
ZPDJVHLHIVCBBN
|
6.3 | IC50 | 3 | — | |
ZTASYFQODPYQIW
|
6.3 | IC50 | 4 | — | |
ZTUNVYDNGSGYLT
|
6.3 | IC50 | 4 | — | |
DFJSJLGUIXFDJP
|
6.2 | Kd | 9 | — | |
HHFBDROWDBDFBR
|
6.2 | Kd | 40 | Yes | |
RXNGGTYNZUEFOM
|
6.2 | IC50 | 8 | Yes | |
KTEIFNKAUNYNJU
|
6.2 | Kd | 114 | — | |
HKKYOSCAKSXOJA
|
6.2 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
RERCSHBOJZUUMN
|
6.2 | IC50 | 2 | — | |
VCZDFACOFNRTMG
|
6.2 | IC50 | 6 | — | |
FOEQINTXCQEBGE
|
6.2 | IC50 | 2 | — | |
FRHDZWLQTMKUPC
|
6.2 | IC50 | 11 | Yes | |
MRZVUZUMBCEAGI
|
6.2 | IC50 | 12 | Yes | |
KOICAHGTHMWKIZ
|
6.2 | IC50 | 6 | Yes | |
VBUMOGXFBGYXDV
|
6.2 | IC50 | 11 | Yes | |
FVPBLAKABVRLRX
|
6.2 | IC50 | 9 | Yes | |
WKDACQVEJIVHMZ
|
6.2 | Kd | 46 | — | |
AULCRCVNIWNUTH
|
6.2 | IC50 | 10 | Yes | |
CJXUHPRULWSPBE
|
6.2 | IC50 | 7 | — | |
BCTIPSBBPQBXAG
|
6.2 | IC50 | 4 | — | |
JVAFTPDILUBIGR
|
6.2 | IC50 | 7 | — | |
JMGXJHWTVBGOKG
|
6.2 | Kd | 7 | — | |
HHZIURLSWUIHRB
|
6.1 | Kd | 57 | Yes | |
KUUKOPMICNKRGE
|
6.1 | IC50 | 12 | Yes | |
LCQAIZAFSOZWRC
|
6.1 | IC50 | 8 | Yes | |
LETIJBVXDGOQFG
|
6.1 | IC50 | 5 | — | |
QQWUGDVOUVUTOY
|
6.1 | Kd | 231 | Yes | |
ZHBTZVAVYLOIKW
|
6.1 | IC50 | 11 | Yes | |
GEPKFPGFWUHVLZ
|
6.1 | IC50 | 6 | Yes | |
JVAFTPDILUBIGR
|
6.1 | IC50 | 9 | Yes | |
JBMGNUFDDDRKSW
|
6.1 | IC50 | 6 | Yes | |
PIOFIWWMFVHCRR
|
6.1 | IC50 | 2 | — | |
SRCAIQMBBDVLGX
|
6.1 | IC50 | 3 | Yes | |
FASPJDRKOSUHHS
|
6.1 | IC50 | 10 | Yes | |
MRZVUZUMBCEAGI
|
6.0 | IC50 | 11 | Yes | |
MVCOAUNKQVWQHZ
|
6.0 | IC50 | 54 | Yes | |
ABQLLFONNKQLLB
|
6.0 | IC50 | 4 | — |