Target Details
| UniProt AC | P54760 |
|---|---|
| Gene Symbol | EPHB4 |
| Protein Name | Ephrin type-B receptor 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 533
- Clinical molecules 99
- Avg pChEMBL 6.88
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (533)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DEMGLABBZSLUOH
|
9.9 | IC50 | 3 | — | |
WYMDWWZXERLYKQ
|
9.8 | IC50 | 3 | — | |
MLDQJTXFUGDVEO
|
9.7 | IC50 | 85 | Yes | |
MXEHLGSSZLWMBO
|
9.6 | IC50 | 3 | — | |
XLBQFFPUVVTFGK
|
9.6 | IC50 | 3 | — | |
FZQWDHPNNCNJFX
|
9.5 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
9.5 | Kd | 102 | Yes | |
CASSAPBDIVDPCC
|
9.4 | IC50 | 3 | Yes | |
GXCMCDVHMWZWJF
|
9.4 | IC50 | 2 | — | |
INFKEXSACBWFSL
|
8.9 | IC50 | 2 | — | |
MPAZWMVMQVIHKE
|
8.8 | IC50 | 2 | — | |
VZHPNWDSQYCLOK
|
8.7 | IC50 | 3 | — | |
GQWMMMAUWHLIBA
|
8.7 | IC50 | 2 | — | |
MIIRGIJHJBFFEA
|
8.5 | IC50 | 3 | — | |
JYLMIXWMBBGQSD
|
8.5 | IC50 | 3 | — | |
QLFGDTPACJHLRY
|
8.5 | IC50 | 3 | — | |
LGYDLRSRBICQTP
|
8.4 | IC50 | 3 | Yes | |
IXIJKXSIADDKHR
|
8.4 | IC50 | 12 | — | |
ZCCPLJOKGAACRT
|
8.4 | IC50 | 599 | — | |
KMKFPXBYIRFWKQ
|
8.3 | IC50 | 3 | Yes | |
VDJMIERKUPUGPE
|
8.3 | IC50 | 3 | — | |
DSRUNANRDDLTEB
|
8.3 | IC50 | 9 | — | |
BETBNWGUKZUUAX
|
8.3 | IC50 | 21 | — | |
JTWMOWRMSZZHDR
|
8.3 | IC50 | 13 | — | |
PPAUQWVFTKFTKY
|
8.3 | IC50 | 3 | Yes | |
ZHMCGBRGDVCXLS
|
8.3 | IC50 | 5 | — | |
IVWHSTCJCURGMH
|
8.2 | IC50 | 2 | — | |
BUHNODQEWUMKMH
|
8.2 | IC50 | 4 | Yes | |
HVQYZYIFVKBRGI
|
8.1 | IC50 | 3 | — | |
URNMUIDFWOJTPW
|
8.1 | Ki | 7 | Yes | |
IVXGFXACZQBKSB
|
8.1 | IC50 | 2 | — | |
DLGLTPBGHQDZCX
|
8.1 | IC50 | 3 | — | |
XTPVNGSRCXLMPE
|
8.1 | IC50 | 3 | — | |
HLXNWJIVTARMJY
|
8.1 | IC50 | 3 | Yes | |
NEJHRDWZMTYHKT
|
8.0 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
8.0 | Kd | 130 | Yes | |
LQSGDXCDNZWTJN
|
8.0 | IC50 | 17 | — | |
HVLNVFOAUCUYQK
|
7.9 | IC50 | 3 | Yes | |
OOZBLQPABHWRKB
|
7.9 | IC50 | 3 | — | |
SEJGTFPOEJWEGG
|
7.9 | Kd | 149 | — | |
VAARYSWULJUGST
|
7.9 | Kd | 119 | Yes | |
FWWFUGDJLTVEBU
|
7.9 | IC50 | 3 | Yes | |
FCCZSKATTXDLOB
|
7.8 | IC50 | 3 | Yes | |
RIXPLQXGEZCOTA
|
7.8 | IC50 | 3 | Yes | |
DNZYFEKYHPAIRX
|
7.8 | IC50 | 3 | — | |
GHGWDSZSHZNVLE
|
7.8 | IC50 | 3 | Yes | |
JGISZYJIPFCGCZ
|
7.8 | IC50 | 3 | — | |
AQSSMEORRLJZLU
|
7.8 | IC50 | 34 | Yes | |
VPZJPWYTYAAMDI
|
7.8 | IC50 | 3 | Yes | |
QYPSALIXKCRYNZ
|
7.8 | IC50 | 12 | Yes |