Target Details
| UniProt AC | P54756 |
|---|---|
| Gene Symbol | EPHA5 |
| Protein Name | Ephrin type-A receptor 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 35
- Clinical molecules 11
- Avg pChEMBL 7.05
KEGG Pathways (1)
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBNZXTGUTAYRHI
|
9.6 | Kd | 102 | Yes | |
AQSSMEORRLJZLU
|
9.4 | Kd | 34 | Yes | |
JTWMOWRMSZZHDR
|
8.5 | IC50 | 13 | — | |
SFCBIFOAGRZJNX
|
8.5 | Kd | 22 | — | |
SEJGTFPOEJWEGG
|
8.2 | Kd | 149 | — | |
PHXJVRSECIGDHY
|
8.1 | Kd | 59 | — | |
ZCCPLJOKGAACRT
|
8.0 | IC50 | 599 | — | |
VAARYSWULJUGST
|
7.8 | Kd | 119 | Yes | |
YOBIWCLAYQWPPW
|
7.6 | IC50 | 23 | — | |
UBPYILGKFZZVDX
|
7.6 | Kd | 130 | Yes | |
CXQHYVUVSFXTMY
|
7.4 | Kd | 154 | — | |
DKZYXHCYPUVGAF
|
7.1 | Kd | 112 | — | |
ALKJNCZNEOTEMP
|
7.1 | Kd | 55 | — | |
XKFTZKGMDDZMJI
|
7.1 | Kd | 64 | Yes | |
MVCOAUNKQVWQHZ
|
7.0 | IC50 | 54 | Yes | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 213 | — | |
ODPGGGTTYSGTGO
|
6.8 | Kd | 153 | — | |
UQRCJCNVNUFYDX
|
6.7 | Kd | 27 | — | |
UHTHHESEBZOYNR
|
6.6 | Kd | 66 | Yes | |
OMZCMEYTWSXEPZ
|
6.6 | Kd | 43 | Yes | |
MWKSRKSEWLRPBL
|
6.5 | IC50 | 1075 | — | |
ZGBAJMQHJDFTQJ
|
6.5 | Kd | 15 | — | |
MLDQJTXFUGDVEO
|
6.4 | Kd | 85 | Yes | |
DKNUPRMJNUQNHR
|
6.4 | Kd | 33 | — | |
WKDACQVEJIVHMZ
|
6.3 | Kd | 46 | — | |
SPMVMDHWKHCIDT
|
6.2 | Kd | 30 | — | |
AAKJLRGGTJKAMG
|
6.2 | Kd | 50 | Yes | |
WVUNYSQLFKLYNI
|
6.2 | Kd | 46 | Yes | |
DFJSJLGUIXFDJP
|
6.1 | Kd | 9 | — | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KTEIFNKAUNYNJU
|
6.0 | Kd | 114 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |