Target Details
| UniProt AC | P54753 |
|---|---|
| Gene Symbol | EPHB3 |
| Protein Name | Ephrin type-B receptor 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 25
- Clinical molecules 7
- Avg pChEMBL 7.12
KEGG Pathways (1)
Active Molecules (25)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AQSSMEORRLJZLU
|
8.7 | Kd | 34 | Yes | |
ZCCPLJOKGAACRT
|
8.2 | IC50 | 599 | — | |
ZBNZXTGUTAYRHI
|
8.2 | Kd | 102 | Yes | |
CCLATZMUQLEESJ
|
8.2 | IC50 | 2 | — | |
XSNFPLSUBIEKQI
|
8.2 | IC50 | 3 | — | |
ZHMCGBRGDVCXLS
|
8.2 | IC50 | 5 | — | |
JTWMOWRMSZZHDR
|
7.8 | IC50 | 13 | — | |
KBWZVVPCJMAFMN
|
7.8 | IC50 | 3 | — | |
AIKGYQDFIJRQIY
|
7.7 | IC50 | 9 | — | |
PCSKFQHKWWNIKM
|
7.3 | IC50 | 7 | — | |
DGSMEFWSLXFLQA
|
7.1 | IC50 | 2 | — | |
SFCBIFOAGRZJNX
|
7.1 | Kd | 22 | — | |
CXQHYVUVSFXTMY
|
7.1 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.1 | Kd | 149 | — | |
XKFTZKGMDDZMJI
|
6.8 | Kd | 64 | Yes | |
MWKSRKSEWLRPBL
|
6.7 | IC50 | 1075 | — | |
UBPYILGKFZZVDX
|
6.7 | Kd | 130 | Yes | |
VAARYSWULJUGST
|
6.5 | Kd | 119 | Yes | |
YMSXHRWUGLAAKL
|
6.5 | IC50 | 14 | Yes | |
PHXJVRSECIGDHY
|
6.3 | Kd | 59 | — | |
HKSZLNNOFSGOKW
|
6.1 | IC50 | 408 | — | |
HHZIURLSWUIHRB
|
6.0 | Kd | 57 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |