Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WIOSRHGIFUMFNQ
|
7.0 | IC50 | 3 | — | |
JVGYDVFOXCBHRN
|
7.0 | IC50 | 3 | — | |
LNELWUPBSLZUIQ
|
7.0 | IC50 | 3 | — | |
OMNGIUDHDBCZAD
|
7.0 | IC50 | 3 | — | |
RZEYZCLEVMBHDS
|
7.0 | IC50 | 3 | — | |
VELNJFTUSCXPKE
|
7.0 | IC50 | 3 | — | |
VERYSPNRLYNKET
|
7.0 | IC50 | 3 | — | |
XEGYXYUUSUWLRL
|
7.0 | IC50 | 3 | — | |
FMHKZUBBRRVRLJ
|
7.0 | IC50 | 3 | — | |
LEQLMZLBAGAUDL
|
7.0 | IC50 | 3 | — | |
DKRDXFRQADAIHU
|
7.0 | IC50 | 3 | — | |
DOTFZTSFGIKARD
|
7.0 | IC50 | 3 | — | |
KVMXASWJIZJMBZ
|
7.0 | IC50 | 3 | — | |
PBXYUGSYGCBAKT
|
7.0 | IC50 | 3 | — | |
ACZBEPYVSHJPFB
|
7.0 | IC50 | 3 | — | |
BSSGJYYHYVLYMA
|
7.0 | IC50 | 3 | — | |
FVVVRFIRYVUVEI
|
7.0 | IC50 | 3 | — | |
IXQRCVAKBIMUJN
|
7.0 | IC50 | 3 | — | |
TYMBPQQASYCWEH
|
7.0 | IC50 | 3 | — | |
XXIPRLNKXMMFIK
|
7.0 | IC50 | 3 | — | |
GLUMAFSYFKCMND
|
6.9 | IC50 | 3 | — | |
JTROLECZHRVLFM
|
6.9 | IC50 | 3 | — | |
KHCSAUOHEOUDEI
|
6.9 | IC50 | 3 | — | |
VWDZYEFJJSYZME
|
6.9 | IC50 | 3 | — | |
ZVDAZHCIEJDXMC
|
6.9 | IC50 | 3 | — | |
ANGLWHGRWFOZSQ
|
6.9 | IC50 | 3 | — | |
ZILNXTHNKXUETP
|
6.9 | IC50 | 3 | — | |
KIFHGJKUXDTDBI
|
6.9 | IC50 | 3 | — | |
ZZXWQIDOSVIHIM
|
6.9 | IC50 | 3 | — | |
IAAHGVIRZIKPHA
|
6.9 | IC50 | 3 | — | |
PZHZVFDPQAUVKV
|
6.9 | IC50 | 3 | — | |
PZHZVFDPQAUVKV
|
6.9 | IC50 | 3 | — | |
FWAXXZSYYYRIBS
|
6.8 | IC50 | 3 | — | |
GDQVLYVPAWKIKI
|
6.8 | IC50 | 3 | — | |
JRLDYTVCZWOPME
|
6.8 | IC50 | 3 | — | |
OKGINEWBFLWKOX
|
6.8 | IC50 | 3 | — | |
PNGBBNJWUZFNIY
|
6.8 | IC50 | 3 | — | |
MINIPTTTZPEEKT
|
6.8 | IC50 | 5 | — | |
BZFPDTIGFMRZDI
|
6.8 | IC50 | 3 | — | |
BZFPDTIGFMRZDI
|
6.8 | IC50 | 3 | — | |
MVVQNOPLTGEXNR
|
6.8 | IC50 | 3 | — | |
BZFPDTIGFMRZDI
|
6.8 | IC50 | 3 | — | |
RPFGIRQWMRKNBU
|
6.8 | IC50 | 3 | — | |
YVGRAQYGPYHZDK
|
6.8 | IC50 | 3 | — | |
UDLAXUPVISWZSI
|
6.8 | IC50 | 3 | — | |
CKGZFAMXPLRINR
|
6.8 | IC50 | 3 | — | |
MRQVRXHGMURIIP
|
6.8 | IC50 | 3 | — | |
UASVJHJKCAJGHA
|
6.8 | IC50 | 3 | — | |
ZJUCMUDMRFUTOF
|
6.8 | IC50 | 3 | — | |
BIQGCKNODPBTSC
|
6.8 | IC50 | 3 | — |