Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QWUMEFVSWZCRDK
|
7.7 | IC50 | 3 | — | |
AIKXKABMMRXBQU
|
7.7 | IC50 | 3 | — | |
SKXWAYULKGVUDE
|
7.7 | IC50 | 3 | — | |
TZBBGNNWRKPAEH
|
7.7 | IC50 | 3 | — | |
ZBYZXMQLZZULRF
|
7.7 | IC50 | 3 | — | |
CDWNSXIRMXQPBS
|
7.7 | IC50 | 3 | — | |
HAKBILSEBDWPBF
|
7.7 | IC50 | 3 | — | |
DQKKFAGODSQYOO
|
7.6 | IC50 | 3 | — | |
DTEHKURDWHCADV
|
7.6 | IC50 | 3 | — | |
SBMPCNJJGZDPRT
|
7.6 | IC50 | 3 | — | |
SHRITIDUUZZEIX
|
7.6 | IC50 | 3 | — | |
SJDHGTJKQKPRAR
|
7.6 | IC50 | 3 | — | |
XUAILHHYTLESDG
|
7.6 | IC50 | 3 | — | |
RZUPDLGZAIZBKU
|
7.6 | IC50 | 3 | — | |
AXEQFCFNPOGNCH
|
7.6 | IC50 | 3 | — | |
LOZUTDKVJLMDTB
|
7.6 | IC50 | 3 | — | |
MXNGXYQZCMFPJD
|
7.6 | IC50 | 3 | — | |
QIWVSVNHRDQBOW
|
7.6 | IC50 | 3 | — | |
HAKBILSEBDWPBF
|
7.6 | IC50 | 3 | — | |
POAGQXNCSDVZDH
|
7.6 | IC50 | 3 | — | |
CXGJWWJDXYZFFZ
|
7.6 | IC50 | 3 | — | |
FOZFBBKUKXGMND
|
7.6 | IC50 | 6 | — | |
GJZNHSHBNVLOAO
|
7.6 | IC50 | 3 | — | |
IBAWDCALOOJODQ
|
7.6 | IC50 | 3 | — | |
JIGCMFQAIKAHMI
|
7.6 | IC50 | 3 | — | |
UNRQWEFTRALILW
|
7.6 | IC50 | 3 | — | |
WFSFSRAGPIZNCC
|
7.6 | IC50 | 3 | — | |
XJADPOFFELMXTA
|
7.6 | IC50 | 3 | — | |
XMJAAWKICASNAA
|
7.5 | IC50 | 3 | — | |
HCLONMUJAHJFIH
|
7.5 | IC50 | 3 | — | |
NRIDLTZEDZLZBY
|
7.5 | IC50 | 3 | — | |
HDOMITVZYCSMIG
|
7.5 | IC50 | 4 | — | |
IONSWNYPWLSPDK
|
7.5 | IC50 | 4 | — | |
KOOPKPXDGQEPLM
|
7.5 | IC50 | 3 | — | |
OIQLBVLVMHTKBC
|
7.5 | IC50 | 4 | — | |
SDTZIRBETDMBLS
|
7.5 | IC50 | 3 | — | |
SGRJQQJTJHBFTK
|
7.5 | IC50 | 3 | — | |
WXGZVKRAYFNMHG
|
7.5 | IC50 | 3 | — | |
CVOILQIVJFYVAQ
|
7.5 | IC50 | 3 | — | |
IRSHUSVLDQPATB
|
7.5 | IC50 | 3 | — | |
NOZMPLJNURLIAQ
|
7.5 | IC50 | 2 | — | |
SVAHBGDAAWZCBA
|
7.5 | IC50 | 3 | — | |
UFODZZUTBCVMAU
|
7.5 | IC50 | 3 | — | |
BXZMPJVMGAVKJS
|
7.5 | IC50 | 3 | — | |
XRYJHUBBBIIQDO
|
7.5 | IC50 | 3 | — | |
YKYCEIQQBDUXHL
|
7.5 | IC50 | 3 | — | |
OKQUCPHNAVGTKM
|
7.4 | IC50 | 3 | — | |
ALQSQGPOANFHOP
|
7.4 | IC50 | 3 | — | |
HTAKTLWSUKQRRS
|
7.4 | IC50 | 3 | — | |
JGQBOOQITKPWJR
|
7.4 | IC50 | 3 | — |