Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PZHZVFDPQAUVKV
|
7.9 | IC50 | 3 | — | |
RVHZRSIRMVWVKL
|
7.9 | IC50 | 3 | — | |
UOVIXKXDBWHQHI
|
7.9 | IC50 | 3 | — | |
YFAHCXPQQYYPCW
|
7.9 | IC50 | 3 | — | |
YTOUKKHZMQVQLZ
|
7.9 | IC50 | 3 | — | |
UFODZZUTBCVMAU
|
7.9 | IC50 | 3 | — | |
DDNCQMVWWZOMLN
|
7.8 | Kd | 2 | — | |
FBPBJZZMBZEJSF
|
7.8 | IC50 | 3 | — | |
IMKYKBMLZRNQRQ
|
7.8 | IC50 | 3 | — | |
IQIUSKXHLPBBOV
|
7.8 | IC50 | 3 | — | |
IVPWVFJBRNZRTL
|
7.8 | IC50 | 3 | — | |
NVHXYCYDLGRUMP
|
7.8 | IC50 | 3 | — | |
PFDYAXRVKURLCH
|
7.8 | IC50 | 3 | — | |
PNGBBNJWUZFNIY
|
7.8 | IC50 | 3 | — | |
PNGBBNJWUZFNIY
|
7.8 | IC50 | 3 | — | |
PUKNFFAMUWZTGI
|
7.8 | IC50 | 3 | — | |
MYYHBCJMEYIHMC
|
7.8 | IC50 | 3 | — | |
PYLSAACWAQSKHB
|
7.8 | IC50 | 3 | — | |
ZPMKSBYSMXCOIZ
|
7.8 | IC50 | 3 | — | |
BHFKZPHEMFPTRO
|
7.8 | IC50 | 3 | — | |
JHGCAWXOMLLFMA
|
7.8 | IC50 | 3 | — | |
LBAWYUCYPDZBSF
|
7.8 | IC50 | 3 | — | |
NDQZTZXQHDYXCS
|
7.8 | IC50 | 3 | — | |
OSHMEGNKNUJDSU
|
7.8 | IC50 | 3 | — | |
OUZGHMLKYZAFHY
|
7.8 | IC50 | 3 | — | |
JWCLZUXPDRRRJM
|
7.8 | IC50 | 3 | — | |
RTFUGASLKHCGCN
|
7.8 | IC50 | 3 | — | |
SFHHXFFUCFPQDI
|
7.8 | IC50 | 3 | — | |
ZIOQYWFVMVDZRK
|
7.8 | IC50 | 3 | — | |
FDEJYPFAUDLEJD
|
7.7 | IC50 | 3 | — | |
FTOYLOIRXWDMMT
|
7.7 | IC50 | 3 | — | |
HUQJJAUBVULGLS
|
7.7 | IC50 | 3 | — | |
MXRHKEUIFABQMB
|
7.7 | IC50 | 3 | — | |
POVOCAKFKAXGDL
|
7.7 | IC50 | 3 | — | |
QKGSYYLRVJDNCK
|
7.7 | IC50 | 3 | — | |
QLFKDVQWAWXRKU
|
7.7 | IC50 | 3 | — | |
SIHCYERWXIEFJJ
|
7.7 | IC50 | 3 | — | |
UJDVXLMRTWCGAG
|
7.7 | IC50 | 3 | — | |
USWMJZZZYCJYJT
|
7.7 | IC50 | 3 | — | |
XEBJMVLHZBRKST
|
7.7 | IC50 | 3 | — | |
YBSFEKXKZHHHNB
|
7.7 | IC50 | 3 | — | |
YSJUCDCNAYRULZ
|
7.7 | IC50 | 3 | — | |
JOFWPJKNNJOGJF
|
7.7 | IC50 | 3 | — | |
RWTZKAWRGHZQKR
|
7.7 | IC50 | 3 | — | |
XOLCNKIFKJXEDO
|
7.7 | IC50 | 3 | — | |
HBRGVUVPCCNRAT
|
7.7 | IC50 | 3 | — | |
KZFHUILKKFVOMB
|
7.7 | IC50 | 4 | — | |
NACHXCODXOLYLO
|
7.7 | IC50 | 3 | — | |
PZHZVFDPQAUVKV
|
7.7 | IC50 | 3 | — | |
YGFHMMKTVSGDPM
|
7.7 | IC50 | 3 | — |