Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RPWGRSSYQVYHBU
|
8.1 | IC50 | 3 | — | |
FZNRRDYXYQYTOQ
|
8.1 | IC50 | 3 | — | |
GPZPPQFWVLHHBU
|
8.1 | IC50 | 3 | — | |
LWOWQQZYEXAZTD
|
8.1 | IC50 | 3 | — | |
HUAHNRHWFFYRAT
|
8.0 | IC50 | 3 | — | |
QLVIOCVYPVUMNY
|
8.0 | IC50 | 3 | — | |
FWBNMGXZQLQVCM
|
8.0 | IC50 | 3 | — | |
GUZUXYPWYDLGJF
|
8.0 | IC50 | 3 | — | |
GUZUXYPWYDLGJF
|
8.0 | IC50 | 3 | — | |
WUVAZFJCZQZLEV
|
8.0 | IC50 | 3 | — | |
YDCVOKZJZPJMKM
|
8.0 | IC50 | 3 | — | |
SJDHGTJKQKPRAR
|
8.0 | IC50 | 3 | — | |
VGHIZNBWVGBFNE
|
8.0 | IC50 | 3 | — | |
CBOOBJUJEUVRPS
|
8.0 | IC50 | 3 | — | |
CXKLITMBWWCPKO
|
8.0 | IC50 | 2 | — | |
DHKCBVLJHGLBIR
|
8.0 | IC50 | 3 | — | |
FIIDAEWKLGRESO
|
8.0 | IC50 | 3 | — | |
HBPSFVFPHQLJNX
|
8.0 | IC50 | 3 | — | |
HGDYRQQUYCUFTK
|
8.0 | IC50 | 4 | — | |
JKKDCZMQLGLGTR
|
8.0 | IC50 | 4 | — | |
KQRMPLPRESELFZ
|
8.0 | IC50 | 4 | — | |
ZCARSOPJYGJCRQ
|
8.0 | IC50 | 3 | — | |
DEUYOHGQAHRUAK
|
8.0 | IC50 | 3 | — | |
DPLDHHPOPUXGGW
|
8.0 | IC50 | 3 | — | |
JCJMWMYJXUGFNN
|
8.0 | IC50 | 3 | — | |
LYTFVMCVYKXNKM
|
8.0 | IC50 | 3 | — | |
LYTFVMCVYKXNKM
|
8.0 | IC50 | 3 | — | |
MDKARWWQHZIIKR
|
8.0 | IC50 | 3 | — | |
NAPUFLNYEBBQPU
|
8.0 | IC50 | 3 | — | |
NAPUFLNYEBBQPU
|
8.0 | IC50 | 3 | — | |
NPLKFZSTTQLUHS
|
8.0 | IC50 | 3 | — | |
RKVBYUMNPKGITG
|
8.0 | IC50 | 3 | — | |
VTULNMARMGUDCN
|
8.0 | IC50 | 3 | — | |
WTKXUHYZWCXYJV
|
8.0 | IC50 | 3 | — | |
XQZACXVVNPRUIZ
|
8.0 | IC50 | 3 | — | |
XXMPIQCOLJGCRH
|
8.0 | IC50 | 3 | — | |
YXAHNICDXLENPY
|
8.0 | IC50 | 3 | — | |
ZJGPWXQIKUCOGR
|
8.0 | IC50 | 3 | — | |
ZJGPWXQIKUCOGR
|
8.0 | IC50 | 3 | — | |
ZPJIMTDAUYYCBN
|
8.0 | IC50 | 3 | — | |
IFZLBONFERYGEE
|
7.9 | IC50 | 3 | — | |
OBFZSUOIZKEKHN
|
7.9 | IC50 | 3 | — | |
MKXYJEZIASGKJZ
|
7.9 | IC50 | 3 | — | |
MSYXYAZMFHMJKN
|
7.9 | IC50 | 3 | — | |
TVGMRVMYCDHOEG
|
7.9 | IC50 | 3 | — | |
YLWZUCCUGZMSMM
|
7.9 | IC50 | 3 | — | |
YORZDHGTKSYMLN
|
7.9 | IC50 | 3 | — | |
BYLOKEGWOSSBIT
|
7.9 | IC50 | 3 | — | |
CQZGCHPJVLXYPV
|
7.9 | IC50 | 3 | — | |
MLGGVHCQGVZWQR
|
7.9 | IC50 | 3 | — |