Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MMFHEXODWCOMFW
|
6.1 | IC50 | 3 | — | |
MUGBFEOWKYVLQV
|
6.1 | IC50 | 3 | — | |
MXQUEDUMKWBYHI
|
6.1 | IC50 | 4 | — | |
ARICWMJJQKCTDR
|
6.1 | IC50 | 3 | — | |
IQMJUBIZVLQDGH
|
6.1 | IC50 | 5 | — | |
PRZKTPKTSVRPRD
|
6.1 | IC50 | 3 | — | |
VFULRIWYLLHLAZ
|
6.1 | IC50 | 10 | — | |
YHCUGGXMFMKHID
|
6.1 | IC50 | 3 | — | |
ZDEYBOGYJCESDB
|
6.1 | IC50 | 2 | — | |
GOAYGCUXFWVPLK
|
6.1 | IC50 | 3 | — | |
ZOSTZZLCBBHOHV
|
6.0 | IC50 | 5 | — | |
DKMMERLAIZECBD
|
6.0 | IC50 | 3 | — | |
JFIAGDXCALKCOT
|
6.0 | IC50 | 4 | — | |
MNLJXFJFDDDISE
|
6.0 | IC50 | 2 | — | |
BKCCUUCEIIWZGH
|
6.0 | IC50 | 3 | — | |
CLKQIZVTONEYRO
|
6.0 | IC50 | 3 | — | |
DXOFVCUNIQMKDW
|
6.0 | IC50 | 4 | — | |
GESSGPHQVIWQGV
|
6.0 | IC50 | 4 | — | |
IJCQPYVFQIZZSO
|
6.0 | IC50 | 4 | — | |
JITUOVWOCIXEEZ
|
6.0 | IC50 | 23 | — | |
JLVYUNCWJCTICJ
|
6.0 | IC50 | 4 | — | |
QEJJXMNBAFWGJK
|
6.0 | IC50 | 3 | — | |
VAZHDIZUYWHZFW
|
6.0 | IC50 | 2 | — | |
ZYCRZKBCOCXUNR
|
6.0 | IC50 | 4 | — |