Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UXZFMELJCXGOCQ
|
6.3 | IC50 | 3 | — | |
LXIXZJSFHDNFEZ
|
6.3 | IC50 | 2 | — | |
ZMTDJXQCSYULBW
|
6.3 | IC50 | 3 | — | |
BNRNXUUZRGQAQC
|
6.3 | IC50 | 12 | — | |
RQWUWJPTWQLWON
|
6.3 | IC50 | 3 | — | |
CAHURFTWFHHOPU
|
6.3 | IC50 | 3 | — | |
IORIFVGSXLSIDK
|
6.3 | IC50 | 4 | — | |
LIQGIDGFAWHICN
|
6.3 | IC50 | 3 | — | |
QMMVRSQAVADTQB
|
6.3 | IC50 | 4 | — | |
VGVQYQRJRNGUNU
|
6.3 | IC50 | 3 | — | |
ICTYYJZHJNSZFG
|
6.3 | IC50 | 3 | — | |
DAFCUKHUCRIICD
|
6.3 | IC50 | 2 | — | |
GGQMHLLGYDUHDQ
|
6.3 | IC50 | 2 | — | |
KSAWSLXAMPVOHI
|
6.3 | IC50 | 3 | — | |
RQVFLKLHPKLTIO
|
6.3 | IC50 | 3 | — | |
SZOKENQFAYLAJE
|
6.3 | IC50 | 3 | — | |
ODAVXTCJLMTDFI
|
6.2 | IC50 | 2 | — | |
VQYHPUHKYSSEOB
|
6.2 | IC50 | 5 | — | |
TXMZJMRBPNQFRI
|
6.2 | IC50 | 3 | — | |
YKKSPSQELFSSMW
|
6.2 | IC50 | 3 | — | |
KILJJPMNQOHZIY
|
6.2 | IC50 | 3 | — | |
USXLZPZGBIYQLQ
|
6.2 | IC50 | 3 | — | |
FTTARRILKZGDNU
|
6.2 | IC50 | 5 | — | |
JBTCDZVDBOMRFT
|
6.2 | IC50 | 2 | — | |
YPYKZBZKFWCVCN
|
6.2 | IC50 | 3 | — | |
DFFKHRZBDXKFRH
|
6.2 | IC50 | 4 | — | |
IJXXNTVMDPJVBW
|
6.2 | IC50 | 3 | — | |
ISOFGIBMBLOJRH
|
6.2 | IC50 | 3 | — | |
KPRJCTUCKTYELS
|
6.2 | IC50 | 2 | — | |
RMYFPLHNAGFJMC
|
6.2 | IC50 | 3 | — | |
MZDYWLVQWRQFMV
|
6.2 | IC50 | 4 | — | |
MZOCQVQIWJPCHX
|
6.2 | IC50 | 2 | — | |
VORFALUWTZNDEJ
|
6.2 | IC50 | 3 | — | |
HIAMRTZPJJKUES
|
6.2 | IC50 | 2 | — | |
MVVQNOPLTGEXNR
|
6.2 | IC50 | 3 | — | |
MVVQNOPLTGEXNR
|
6.2 | IC50 | 3 | — | |
ZCVGFCXGAGKYHH
|
6.2 | IC50 | 3 | — | |
IHPVHEUBCHVJEQ
|
6.2 | IC50 | 2 | — | |
YWZGIRPKPNRMEV
|
6.2 | IC50 | 2 | — | |
ZKSDAVPQRBAJOA
|
6.2 | IC50 | 4 | — | |
OSBOOFALLQCYDR
|
6.2 | IC50 | 3 | — | |
WSLKNNDWDHGJQK
|
6.2 | IC50 | 2 | — | |
XRIYYPDCPKIHRW
|
6.2 | IC50 | 3 | — | |
FXUFWAVOAYRFKB
|
6.2 | IC50 | 5 | — | |
LWAQPJWARNOJEY
|
6.1 | IC50 | 3 | — | |
IVICMAQJTMYPDI
|
6.1 | IC50 | 2 | — | |
JTROLECZHRVLFM
|
6.1 | IC50 | 3 | — | |
UBXCQPGYHRWIKD
|
6.1 | IC50 | 3 | — | |
ALVRWLFAONYUAV
|
6.1 | IC50 | 3 | — | |
DDKCZVDGSHWYON
|
6.1 | IC50 | 4 | — |