Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BFFSRRAKFFTYRB
|
6.5 | IC50 | 3 | — | |
XKHNGFDZRPJTCY
|
6.5 | IC50 | 3 | — | |
YRRWQMBIMZMVDB
|
6.5 | IC50 | 4 | — | |
PZKOOBRKCGIRJF
|
6.5 | IC50 | 3 | — | |
AQLHITNAEZNQJK
|
6.5 | IC50 | 3 | — | |
AQLHITNAEZNQJK
|
6.5 | IC50 | 3 | — | |
CEASKHHYUJNGEA
|
6.5 | IC50 | 3 | — | |
ORDCDFJDRJJITQ
|
6.5 | IC50 | 5 | — | |
QVDZHWJXZYVABG
|
6.5 | IC50 | 3 | — | |
LXIXZJSFHDNFEZ
|
6.5 | IC50 | 3 | — | |
MZDJCPNZHVQURG
|
6.5 | IC50 | 3 | — | |
PDEQSHWWQUGZQW
|
6.5 | IC50 | 3 | — | |
RPFGNHZGIBGJKF
|
6.5 | IC50 | 2 | — | |
UXZFMELJCXGOCQ
|
6.5 | IC50 | 2 | — | |
GEKRVCRUZXROSZ
|
6.5 | IC50 | 3 | — | |
GEKRVCRUZXROSZ
|
6.5 | IC50 | 3 | — | |
OFZGCAMFVYIIHV
|
6.5 | IC50 | 24 | — | |
PZKOOBRKCGIRJF
|
6.5 | IC50 | 3 | — | |
LEYPTBGWIKQYRW
|
6.5 | IC50 | 3 | — | |
LEYPTBGWIKQYRW
|
6.5 | IC50 | 3 | — | |
LEYPTBGWIKQYRW
|
6.5 | IC50 | 3 | — | |
YXOLEIZBMQWRJW
|
6.5 | IC50 | 3 | — | |
OAFVIHQZGHZRRA
|
6.5 | IC50 | 2 | — | |
NSFYZWGFIIQKQP
|
6.4 | IC50 | 3 | — | |
BEWJVJUTJZTWQQ
|
6.4 | IC50 | 3 | — | |
IZGDUNLRMAOQTD
|
6.4 | IC50 | 4 | — | |
KLXXAXDPPNWJOU
|
6.4 | IC50 | 2 | — | |
CNYPMSYZXANIAK
|
6.4 | IC50 | 4 | — | |
BNYIEPJRYJQTHM
|
6.4 | IC50 | 2 | — | |
CXGGCYJPLGSTBH
|
6.4 | IC50 | 3 | — | |
HWZIGTUHYHCMIT
|
6.4 | IC50 | 3 | — | |
KJNDGYWAQRWMBO
|
6.4 | IC50 | 3 | — | |
KAIFDCSXZCWWKF
|
6.4 | IC50 | 3 | — | |
UBSAKYMRJJOZDY
|
6.4 | IC50 | 3 | — | |
KYLSIDIKSXHHCI
|
6.4 | IC50 | 3 | — | |
OYBSUAILVMFPHS
|
6.4 | IC50 | 3 | — | |
RVWGYNGTLDYNPU
|
6.4 | IC50 | 3 | — | |
XFUMOUGBVYWUFH
|
6.4 | IC50 | 3 | — | |
APQLMNUUGPWXRZ
|
6.4 | IC50 | 3 | — | |
OSXMMCYBFRYLSU
|
6.4 | IC50 | 3 | — | |
WBJONNSPSBKOSD
|
6.4 | IC50 | 5 | — | |
ARZYUJKMHFQSRW
|
6.3 | IC50 | 3 | — | |
BPTCRJBPJDAUBH
|
6.3 | IC50 | 3 | — | |
BRAWZTIBDHEBNS
|
6.3 | IC50 | 3 | — | |
HCLWEXNPZAAMRB
|
6.3 | IC50 | 3 | — | |
HIAMRTZPJJKUES
|
6.3 | IC50 | 2 | — | |
JBTCDZVDBOMRFT
|
6.3 | IC50 | 3 | — | |
SQYNPZYBHGTSOY
|
6.3 | IC50 | 5 | — | |
XQZOCZINLVECTD
|
6.3 | IC50 | 2 | — | |
QRWHTFXNHZLJAL
|
6.3 | IC50 | 5 | — |