Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKFYCHHMKLLPQY
|
6.8 | IC50 | 3 | — | |
IVIOKHSMYSCNPJ
|
6.7 | IC50 | 3 | — | |
RZZDUEKLZBHEJJ
|
6.7 | IC50 | 3 | — | |
GRFJYHDUOKDAKO
|
6.7 | IC50 | 3 | — | |
LWKMAOPQFDSIHC
|
6.7 | IC50 | 3 | — | |
NSFYZWGFIIQKQP
|
6.7 | IC50 | 3 | — | |
RVJAZKLTOAMCHB
|
6.7 | IC50 | 3 | — | |
AKDKVOQBJMHADC
|
6.7 | IC50 | 3 | — | |
BFXFDLMTMKFDSG
|
6.7 | IC50 | 3 | — | |
DGHWUYQHCWDSCX
|
6.7 | IC50 | 4 | — | |
GOESVWYTXYEMCF
|
6.7 | IC50 | 4 | — | |
MCTQXSSLZDBVEP
|
6.7 | IC50 | 3 | — | |
NYYKSMYMZPDEJH
|
6.7 | IC50 | 3 | — | |
SLLWQPUNKSEVKT
|
6.7 | IC50 | 4 | — | |
SVNBZNOJEMDHHP
|
6.7 | IC50 | 3 | — | |
VCAGHSXTTDHBAV
|
6.7 | IC50 | 3 | — | |
XCOUYJYBUSTRSB
|
6.7 | IC50 | 3 | — | |
SBPLRPBAFIENJD
|
6.7 | IC50 | 3 | — | |
DURMBXZBTJGGSF
|
6.7 | IC50 | 3 | — | |
IOBLPVSVJNVETM
|
6.7 | IC50 | 3 | — | |
SWHFTCTZWOUUQD
|
6.7 | IC50 | 3 | — | |
NHTZYYDADSWQFF
|
6.7 | IC50 | 3 | — | |
SQDRHBKRJBDLOC
|
6.6 | IC50 | 3 | — | |
VRSLRMWKAICODM
|
6.6 | IC50 | 3 | — | |
ZEUKRJZWWLBXIK
|
6.6 | IC50 | 3 | — | |
MVBCAJXPQPBVSA
|
6.6 | IC50 | 3 | — | |
RPFGNHZGIBGJKF
|
6.6 | IC50 | 3 | — | |
XKGOGXSNJQICIE
|
6.6 | IC50 | 3 | — | |
ICFZMMURQAUHKS
|
6.6 | IC50 | 3 | — | |
NOGPVEPEDSPNHF
|
6.6 | IC50 | 3 | — | |
YWWHXMUOPZSUDB
|
6.6 | IC50 | 3 | — | |
YWWHXMUOPZSUDB
|
6.6 | IC50 | 3 | — | |
MNWITQKMYDXVBF
|
6.6 | IC50 | 3 | — | |
HEERUKANWGHTOL
|
6.6 | IC50 | 3 | — | |
MVICHLUMJUWVOO
|
6.6 | IC50 | 3 | — | |
MWKYQHIHOQUVGV
|
6.6 | IC50 | 3 | — | |
VQUWFLFKDYALSX
|
6.6 | IC50 | 3 | — | |
ONUWUZXNTMRHEG
|
6.6 | IC50 | 2 | — | |
SECKRCOLJRRGGV
|
6.6 | IC50 | 16 | — | |
KRADQTILGMSJGT
|
6.6 | IC50 | 2 | — | |
XUHWSBHEGYQEDI
|
6.6 | IC50 | 3 | — | |
AAAZUNCZBZHDPM
|
6.5 | IC50 | 3 | — | |
GMPCYHZOARRAOF
|
6.5 | IC50 | 3 | — | |
HVRCNXOHZPZGSJ
|
6.5 | IC50 | 3 | — | |
MVVQNOPLTGEXNR
|
6.5 | IC50 | 3 | — | |
MVVQNOPLTGEXNR
|
6.5 | IC50 | 3 | — | |
OJTUUGACOKQJNT
|
6.5 | IC50 | 3 | — | |
PHHOODNTGCUZFM
|
6.5 | IC50 | 3 | — | |
YJCZMNIYQABZMT
|
6.5 | IC50 | 3 | — | |
AIVNVMRJLJHFCU
|
6.5 | IC50 | 4 | — |