Target Details
| UniProt AC | P54750 |
|---|---|
| Gene Symbol | PDE1A |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 624
- Clinical molecules 0
- Avg pChEMBL 7.44
KEGG Pathways (7)
Active Molecules (624)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KQMWFBJUYHOBDC
|
10.0 | Ki | 2 | — | |
UJLHNYPXKZJKLV
|
10.0 | IC50 | 24 | — | |
KXCOKRBRUWINCT
|
9.9 | IC50 | 24 | — | |
NIXYLBKMUOTNON
|
9.8 | IC50 | 3 | — | |
NIXYLBKMUOTNON
|
9.8 | IC50 | 3 | — | |
OWQWYQRHXWXXOX
|
9.8 | IC50 | 3 | — | |
KPFFPWNKWSYQFT
|
9.8 | IC50 | 24 | — | |
RKEUHNQOPBPRQD
|
9.7 | Ki | 2 | — | |
YAZFJAWMJDOHDF
|
9.7 | IC50 | 6 | — | |
GOBQSCBEINUNFL
|
9.6 | IC50 | 24 | — | |
KLLVPOPJMWWQFO
|
9.6 | IC50 | 3 | — | |
KSTNYSJSCGBUFA
|
9.6 | IC50 | 6 | — | |
SJMDRHYXKHAMKH
|
9.6 | IC50 | 3 | — | |
ITYGOFCAYSOSFS
|
9.5 | Ki | 2 | — | |
AFCWMWBOATWMJV
|
9.5 | IC50 | 24 | — | |
DKSKKVAOIPURFT
|
9.5 | IC50 | 24 | — | |
GHJOVBRBPVEUOD
|
9.5 | IC50 | 3 | — | |
OQHANCKZXQVDDH
|
9.5 | IC50 | 3 | — | |
OUTHEXWIIRDFDE
|
9.5 | IC50 | 3 | — | |
OUTHEXWIIRDFDE
|
9.5 | IC50 | 3 | — | |
HINKCAKLUHRIQD
|
9.4 | IC50 | 3 | — | |
LOSBPLVFUGTAOA
|
9.4 | IC50 | 3 | — | |
ROWMNTAKQCZGNZ
|
9.4 | IC50 | 3 | — | |
QOYNQFLWGDTXKT
|
9.3 | IC50 | 3 | — | |
HHYVSMVGFQLTLE
|
9.3 | IC50 | 3 | — | |
PSUHAEXBWCRQED
|
9.3 | Ki | 2 | — | |
DBRGOFPEANLZGU
|
9.1 | IC50 | 3 | — | |
DGDYHVXCROBNNK
|
9.1 | IC50 | 3 | — | |
DGDYHVXCROBNNK
|
9.1 | IC50 | 3 | — | |
GHHGVGRPPLMROZ
|
9.1 | IC50 | 3 | — | |
MKELJWFWEJOZNC
|
9.1 | IC50 | 3 | — | |
OZQQLPFSQLZXQT
|
9.1 | IC50 | 3 | — | |
SXNFSKBWTTYFLI
|
9.0 | IC50 | 3 | — | |
XJUDCWZJLDFIBG
|
9.0 | IC50 | 3 | — | |
BPBDCOLBZYWXHD
|
9.0 | IC50 | 24 | — | |
BVKDBZHCRMPMSA
|
9.0 | IC50 | 3 | — | |
DAJMAHYQLJFZEY
|
9.0 | IC50 | 3 | — | |
FIZYUMZEYFRNCJ
|
9.0 | IC50 | 3 | — | |
FLZRLEPPHKZGPK
|
9.0 | IC50 | 3 | — | |
FMMIDZWTNQYEIY
|
9.0 | IC50 | 24 | — | |
SYWOKLNWWYOPHL
|
9.0 | IC50 | 3 | — | |
SYWOKLNWWYOPHL
|
9.0 | IC50 | 3 | — | |
IGMSFVIKHQRGSP
|
9.0 | IC50 | 3 | — | |
LRTCNZDFQQIFPH
|
9.0 | IC50 | 3 | — | |
CJOUFKUESMXTOX
|
8.9 | IC50 | 3 | — | |
DFUHIVBKOGIXKT
|
8.9 | IC50 | 3 | — | |
XOIXJVILDWTHEL
|
8.9 | IC50 | 3 | — | |
XOIXJVILDWTHEL
|
8.9 | IC50 | 3 | — | |
IWDHUHWZRSHWGD
|
8.8 | IC50 | 3 | — | |
JYRPZCKZXZYAOY
|
8.8 | IC50 | 3 | — |