Target Details
| UniProt AC | P54619 |
|---|---|
| Gene Symbol | PRKAG1 |
| Protein Name | 5'-AMP-activated protein kinase subunit gamma-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00571 (CBS) |
Summary
- Multi-target molecules 83
- Clinical molecules 11
- Avg pChEMBL 7.01
KEGG Pathways (16)
- AMPK signaling pathway
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Apelin signaling pathway
- Circadian rhythm
- FoxO signaling pathway
- Glucagon signaling pathway
- Hypertrophic cardiomyopathy
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- Non-alcoholic fatty liver disease
- Oxytocin signaling pathway
- Thermogenesis
- Tight junction
Active Molecules (83)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YJKYSCKYOBZSRV
|
6.7 | Kd | 3 | — | |
HEPDAJRNJBNJAE
|
6.7 | IC50 | 15 | Yes | |
PIVGOZQUWKCUID
|
6.6 | IC50 | 7 | — | |
ZMAJVXKEVISHMQ
|
6.6 | IC50 | 9 | — | |
VCLMLPXAUIQEEM
|
6.6 | IC50 | 7 | — | |
OOQJIJYKWXLQNC
|
6.5 | IC50 | 16 | Yes | |
KOZFSFOOLUUIGY
|
6.5 | Kd | 88 | Yes | |
WKDACQVEJIVHMZ
|
6.5 | Kd | 46 | — | |
GCQRNJUDAAOEJK
|
6.4 | Kd | 3 | — | |
LQVXSNNAFNGRAH
|
6.4 | Kd | 33 | Yes | |
ZXOKHOODFVNZIC
|
6.3 | IC50 | 7 | — | |
CTESJDQKVOEUOY
|
6.3 | Kd | 3 | — | |
CQZOSLVFDRPCFJ
|
6.3 | IC50 | 7 | — | |
SGMHSWUFNYQVBA
|
6.3 | IC50 | 9 | — | |
JBRGOJOHEISXNB
|
6.2 | Kd | 3 | — | |
XGEBOBAOVSOQCV
|
6.2 | IC50 | 10 | — | |
IAYGCINLNONXHY
|
6.2 | Kd | 50 | — | |
WNLKAYDTKKISBN
|
6.2 | IC50 | 7 | — | |
CAWABSRZIMATJO
|
6.2 | IC50 | 9 | — | |
UARVSLPFGRKWQN
|
6.2 | IC50 | 11 | — | |
INGGFDWTZNSBPY
|
6.1 | IC50 | 7 | — | |
MXJMJNRCJKHFPP
|
6.1 | IC50 | 10 | — | |
YFNWWNRZJGMDBR
|
6.1 | Kd | 35 | — | |
NGDYCJGYGAYDIM
|
6.1 | IC50 | 7 | — | |
ZWIGVNWZHBPXNS
|
6.1 | IC50 | 7 | — | |
HRKJFKJZUNJKNU
|
6.1 | IC50 | 10 | — | |
SLEWGGZPOQNVSU
|
6.1 | Kd | 22 | — | |
BUMYTKZYNNGHLL
|
6.0 | IC50 | 7 | — | |
UIARLYUEJFELEN
|
6.0 | Kd | 289 | Yes | |
WWTRFWLRGARRAD
|
6.0 | IC50 | 10 | — | |
SVJBHQPXESBDEQ
|
6.0 | IC50 | 9 | — | |
FCJGMZMSVIAAJU
|
6.0 | IC50 | 9 | — | |
PIQCTGMSNWUMAF
|
6.0 | Kd | 137 | Yes |