Target Details
| UniProt AC | P54619 |
|---|---|
| Gene Symbol | PRKAG1 |
| Protein Name | 5'-AMP-activated protein kinase subunit gamma-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00571 (CBS) |
Summary
- Multi-target molecules 83
- Clinical molecules 11
- Avg pChEMBL 7.01
KEGG Pathways (16)
- AMPK signaling pathway
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Apelin signaling pathway
- Circadian rhythm
- FoxO signaling pathway
- Glucagon signaling pathway
- Hypertrophic cardiomyopathy
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- Non-alcoholic fatty liver disease
- Oxytocin signaling pathway
- Thermogenesis
- Tight junction
Active Molecules (83)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FJNHSBVZTQFKEF
|
9.0 | IC50 | 7 | — | |
JKGJLUCJLNJXKG
|
8.6 | IC50 | 7 | — | |
FCLPVPNWFDOVKL
|
8.4 | Ki | 11 | — | |
LYADGAGFYYXXIO
|
8.3 | IC50 | 82 | — | |
NOMBUNHXDWBICV
|
8.3 | Ki | 11 | — | |
AYCPARAPKDAOEN
|
8.3 | IC50 | 73 | — | |
CXYVYGXMFQSTKH
|
8.2 | IC50 | 7 | — | |
XRDMDDSSWUSOAX
|
8.1 | IC50 | 7 | — | |
FHQXLWCFSUSXBF
|
8.1 | Kd | 3 | — | |
WGWCRXQUBYJTRA
|
8.0 | Ki | 11 | — | |
NXSJMRCTGYTSTK
|
7.9 | Kd | 200 | — | |
MJHBRTGGZYSCHJ
|
7.9 | Kd | 3 | — | |
GKPYSXKYDOSNMQ
|
7.8 | Kd | 3 | — | |
JQJNGAWEMYQJIQ
|
7.8 | Kd | 3 | — | |
OSVUGUHRKMMBSE
|
7.8 | Kd | 170 | — | |
WQUGCKCCOOBUNT
|
7.8 | IC50 | 7 | — | |
LHDKPFSHXFFALR
|
7.7 | IC50 | 7 | — | |
MWKSRKSEWLRPBL
|
7.7 | Kd | 1075 | — | |
VPUNMIRZXILGLE
|
7.7 | Kd | 3 | — | |
QZCUYXGDXFPQEA
|
7.7 | IC50 | 7 | — | |
NTZCHZCFSJZAQG
|
7.7 | IC50 | 7 | — | |
RHWVKZPITKBHLD
|
7.7 | Kd | 3 | — | |
QZIZUCHLAKADOE
|
7.6 | Kd | 3 | — | |
UEFCSGDOOJJXTN
|
7.6 | IC50 | 46 | — | |
MRMDURIHTGUZQI
|
7.5 | IC50 | 7 | — | |
LOLPPWBBNUVNQZ
|
7.5 | Kd | 97 | Yes | |
WDNAXOPVZIEECR
|
7.5 | IC50 | 11 | — | |
JCVIFVYRMKVCDU
|
7.3 | Kd | 3 | — | |
QFWZHKHVYWARIP
|
7.3 | Kd | 3 | — | |
NGFGTMFVWSDFPS
|
7.3 | IC50 | 32 | — | |
OFPXCBKYWWZZGT
|
7.2 | IC50 | 7 | — | |
WMXDIPVFXWNELM
|
7.2 | IC50 | 14 | Yes | |
CSZAJEXPQFERTK
|
7.2 | IC50 | 10 | — | |
JGMADXMPAZATOC
|
7.1 | Kd | 3 | — | |
XKFTZKGMDDZMJI
|
7.1 | Kd | 64 | Yes | |
QFVPMQJTUWDFKR
|
7.0 | Kd | 3 | — | |
XHBVYDAKJHETMP
|
7.0 | IC50 | 24 | Yes | |
DOTGPNHGTYJDEP
|
7.0 | IC50 | 8 | — | |
SLCNIAWQMQCAFR
|
7.0 | IC50 | 8 | — | |
LTLTUJCGZGVBTO
|
7.0 | Kd | 3 | — | |
BPMMMRKHRUQAAY
|
6.9 | IC50 | 7 | — | |
JRKYKAKARRYSSS
|
6.8 | IC50 | 14 | Yes | |
XLFNLJYGUOLEJS
|
6.8 | IC50 | 26 | — | |
DKZYXHCYPUVGAF
|
6.8 | Kd | 112 | — | |
NOGWJYQSYBAMTO
|
6.8 | Kd | 3 | — | |
UDMBCSSLTHHNCD
|
6.8 | Kd | 11 | — | |
HKSZLNNOFSGOKW
|
6.8 | IC50 | 408 | — | |
GZCJKJJWOUAGMR
|
6.7 | Kd | 3 | — | |
LLRSNVNZYTWKPN
|
6.7 | IC50 | 7 | — | |
IUDLPZTURGVXEA
|
6.7 | Kd | 7 | — |