Target Details
| UniProt AC | P54289 |
|---|---|
| Gene Symbol | CACNA2D1 |
| Protein Name | Voltage-dependent calcium channel subunit alpha-2/delta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08473 (VGCC_alpha2) PF00092 (VWA) PF08399 (VWA_N) |
Summary
- Multi-target molecules 234
- Clinical molecules 0
- Avg pChEMBL 6.92
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WKIWZYVELZLXOB
|
6.5 | Ki | 2 | — | |
WSTIUHFTNYABQA
|
6.5 | Ki | 2 | — | |
WXSFJWUCHFZTTH
|
6.5 | Ki | 2 | — | |
XGWWGIXMFTXMJQ
|
6.5 | Ki | 2 | — | |
XJHDXJNNMHSVDG
|
6.5 | Ki | 2 | — | |
XJHDXJNNMHSVDG
|
6.5 | Ki | 2 | — | |
XJNGDIZTERSHCD
|
6.5 | Ki | 2 | — | |
XMQMKCVOYHQFMM
|
6.5 | Ki | 2 | — | |
YLLGDFRXKJITEN
|
6.5 | Ki | 2 | — | |
ZBZACMIGZBMLSQ
|
6.5 | Ki | 2 | — | |
ZCVHLLHRVFCIKQ
|
6.5 | Ki | 2 | — | |
ZQDPPYZTUFYXQP
|
6.5 | Ki | 2 | — | |
ZWHDVUZVJSBQRG
|
6.5 | Ki | 2 | — | |
PVJNWPXQHNFPOR
|
6.5 | IC50 | 3 | — | |
APFIMMRBLUEEJX
|
6.5 | IC50 | 3 | — | |
NTCNYPJNYIBPSC
|
6.5 | IC50 | 3 | — | |
MTACWCHMAADIEZ
|
6.5 | IC50 | 3 | — | |
QLIONHKEMUXUQB
|
6.5 | Ki | 2 | — | |
IWLOXSUFFLVQCV
|
6.4 | Ki | 2 | — | |
QJXZQIYIFNIJIO
|
6.4 | IC50 | 3 | — | |
DXHGSDDDNQXAEJ
|
6.4 | IC50 | 26 | — | |
SZXAWCKROBFQPN
|
6.3 | IC50 | 3 | — | |
RLEMIIBGFDBVBD
|
6.3 | IC50 | 3 | — | |
GGKXNHJATNHIDB
|
6.3 | IC50 | 3 | — | |
RFHHKLHLLXMGOX
|
6.3 | IC50 | 3 | — | |
UZBVUMAEAIQRKF
|
6.2 | IC50 | 4 | — | |
KGQXWNGARPKIIX
|
6.2 | IC50 | 3 | — | |
CHQJWHDWPUGTOO
|
6.2 | Ki | 2 | — | |
DZLGMNWIHGPMMA
|
6.1 | Ki | 2 | — | |
XKDFZZUFCHOVRN
|
6.1 | IC50 | 27 | — | |
LRBRSWLNUGPGBK
|
6.1 | Ki | 2 | — | |
HNBPLGZOUSBZKX
|
6.1 | Ki | 2 | — | |
YCGNFTGPXBAEMC
|
6.0 | Ki | 2 | — | |
QSGMFCUAWLYRRU
|
6.0 | Ki | 2 | — |