Target Details
UniProt ACP54289
Gene SymbolCACNA2D1
Protein NameVoltage-dependent calcium channel subunit alpha-2/delta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF08473 (VGCC_alpha2) PF00092 (VWA) PF08399 (VWA_N)
Summary
  • Multi-target molecules 234
  • Clinical molecules 0
  • Avg pChEMBL 6.92
Top Co-occurrence Targets
Active Molecules (234)
InChIKey pChEMBL Type Targets Clinical
LAAINAAKDMZDHJ 6.5 Ki 2
LHZQSHOTZSBXMT 6.5 Ki 2
LKHGZBCJCIQCLI 6.5 Ki 2
LKMAZENQDJPAOZ 6.5 Ki 2
LRDBTLRFYYQSHO 6.5 Ki 2
LTMDMFAPAHPHAK 6.5 Ki 2
LTMDMFAPAHPHAK 6.5 Ki 2
LYLPBSIHVCVZJN 6.5 Ki 2
LZASFPSWSSXPPA 6.5 Ki 2
MENDFCYVYYBFRD 6.5 Ki 2
MFIHOGLJRPBYIE 6.5 Ki 2
MFQDHZNLWYDSFC 6.5 Ki 2
MFVCDOIXYGRALQ 6.5 Ki 2
MKPRTPUWLYUUAO 6.5 Ki 2
MLLSPSHXJVRFIL 6.5 Ki 2
MLTWOMDQQFOCMD 6.5 IC50 3
NBFFFSSWIDRREJ 6.5 Ki 2
NBOBGWSKDGTTTF 6.5 Ki 2
NMZMEZDYOKXSFP 6.5 Ki 2
NPZWPKSRTQJPHR 6.5 Ki 2
NSAPWHGIQPPHQR 6.5 Ki 2
OAKSTVOUJWQVNC 6.5 Ki 2
OAWHXCORWBSROR 6.5 Ki 2
OAWHXCORWBSROR 6.5 Ki 2
OUAQODABUANYJQ 6.5 Ki 2
PLRRDJAYJPNCQT 6.5 Ki 2
PLRRDJAYJPNCQT 6.5 Ki 2
PNEPGBCHAGDKHQ 6.5 Ki 2
PQNPVPGYGMGILK 6.5 Ki 2
PVIBEZAPXVLWAG 6.5 Ki 2
PVIBEZAPXVLWAG 6.5 Ki 2
PZUBKBDQWUCFBG 6.5 Ki 2
QIQGSCFPOMYFCX 6.5 Ki 2
QLJXGOSUUYOJJV 6.5 Ki 2
QNGRKOMRLIHMHR 6.5 Ki 2
QZTSBVNAYFBWIC 6.5 Ki 2
ROKYHZXDTGMCJT 6.5 Ki 2
ROKYHZXDTGMCJT 6.5 Ki 2
RPJMFEMGOQFHBY 6.5 Ki 2
RUZCAHKGJLXNSF 6.5 Ki 2
RXAFOXHLNBBCQQ 6.5 Ki 2
SMXRDTCWJPEFLL 6.5 Ki 2
SOALXNOFBIRPAX 6.5 Ki 2
SVLCJDSHPQXKRN 6.5 Ki 2
TUYHONFAVFQREZ 6.5 Ki 2
UYKJZILKOZJTOW 6.5 Ki 2
UYQPTSPEQOJDJK 6.5 Ki 2
UYQPTSPEQOJDJK 6.5 Ki 2
VHLVLBGGLGNCMM 6.5 Ki 2
WCUWYYWDWUAFDE 6.5 Ki 2
2D structure