Target Details
| UniProt AC | P54289 |
|---|---|
| Gene Symbol | CACNA2D1 |
| Protein Name | Voltage-dependent calcium channel subunit alpha-2/delta-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08473 (VGCC_alpha2) PF00092 (VWA) PF08399 (VWA_N) |
Summary
- Multi-target molecules 234
- Clinical molecules 0
- Avg pChEMBL 6.92
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDPXETVZRHNLTM
|
7.5 | IC50 | 3 | — | |
GPVQFLNMUGKFCX
|
7.5 | IC50 | 2 | — | |
IXSXSOMMKYUETH
|
7.5 | IC50 | 26 | — | |
UXTXHFYVRKEMAW
|
7.5 | IC50 | 2 | — | |
FFLKWIPCJQAAJX
|
7.4 | IC50 | 26 | — | |
QRGMHEOPAKSEPT
|
7.4 | IC50 | 26 | — | |
UMDPFCNSBNGNBU
|
7.4 | IC50 | 26 | — | |
IARAKTOMNMLDLY
|
7.4 | IC50 | 4 | — | |
QUDJCWKOPXBSPH
|
7.4 | IC50 | 3 | — | |
QWTOYMMBYIZUDZ
|
7.4 | IC50 | 26 | — | |
AOQSRDPSBXFFQW
|
7.3 | IC50 | 3 | — | |
ROOQZCIZDJRFFY
|
7.3 | IC50 | 3 | — | |
ZWJKOWFFHJCZRL
|
7.3 | IC50 | 26 | — | |
GEHGVVUONLLQIR
|
7.2 | IC50 | 2 | — | |
CNSYGZOEIHDOQH
|
7.2 | IC50 | 3 | — | |
XNUZTIQWJMXUHN
|
7.2 | IC50 | 26 | — | |
AZSLSVQTOKQPLV
|
7.2 | IC50 | 26 | — | |
BQQHWRLQVWTKDU
|
7.1 | IC50 | 26 | — | |
QKEPYKVCOWFCDP
|
7.1 | IC50 | 26 | — | |
JWHAZXDKSGAIEK
|
7.0 | IC50 | 4 | — | |
CCSYRVYORQUIJU
|
7.0 | Ki | 2 | — | |
RTFHWULQHQDWPK
|
7.0 | IC50 | 26 | — | |
GTSIUFNWVXFHJS
|
7.0 | IC50 | 3 | — | |
AOQSRDPSBXFFQW
|
7.0 | IC50 | 4 | — | |
CEXBUHRJNQKOBZ
|
7.0 | IC50 | 3 | — | |
JDFLEUYRGZPZQD
|
7.0 | IC50 | 3 | — | |
VCPMZDWBEWTGNW
|
7.0 | IC50 | 3 | — | |
AOQSRDPSBXFFQW
|
6.8 | IC50 | 3 | — | |
FMJSSIYEDJFGBC
|
6.8 | IC50 | 3 | — | |
PPVBMJIAJXVQFX
|
6.8 | IC50 | 3 | — | |
ZMRQKZANSRISRS
|
6.8 | IC50 | 3 | — | |
POPQMMOUZVBXFY
|
6.8 | IC50 | 3 | — | |
JJWWPFHYFYVBMO
|
6.7 | IC50 | 3 | — | |
RPLRXHLXRQIHHQ
|
6.7 | IC50 | 3 | — | |
YYMGRGSETHUACY
|
6.7 | IC50 | 3 | — | |
JKAOGJXEFQNYHE
|
6.7 | IC50 | 2 | — | |
UQEYHZANEBZUSS
|
6.7 | IC50 | 4 | — | |
PSEHTODILBVIHC
|
6.6 | IC50 | 4 | — | |
CBDZLOJIUYHCHO
|
6.6 | IC50 | 4 | — | |
NIMFDABOPDBIHU
|
6.6 | IC50 | 3 | — | |
HWGMUVSZGFXYSD
|
6.6 | IC50 | 3 | — | |
SFDCNWPOHFHZDB
|
6.6 | Ki | 2 | — | |
DKVOGZPCCPBBPU
|
6.6 | IC50 | 3 | — | |
JCEFNPWMPAOQID
|
6.6 | IC50 | 4 | — | |
QXNYWQVYZYCACA
|
6.6 | IC50 | 3 | — | |
KGKFKQGQYIUQAL
|
6.6 | IC50 | 3 | — | |
DOVZOQYQXHNCCN
|
6.5 | IC50 | 3 | — | |
YZBMBXSAQFTDCP
|
6.5 | IC50 | 3 | — | |
ADZLFOZXVROIJQ
|
6.5 | Ki | 2 | — | |
AMKWNLRAFBRBBP
|
6.5 | Ki | 2 | — |