Target Details
UniProt ACP54289
Gene SymbolCACNA2D1
Protein NameVoltage-dependent calcium channel subunit alpha-2/delta-1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF08473 (VGCC_alpha2) PF00092 (VWA) PF08399 (VWA_N)
Summary
  • Multi-target molecules 234
  • Clinical molecules 0
  • Avg pChEMBL 6.92
Top Co-occurrence Targets
Active Molecules (234)
InChIKey pChEMBL Type Targets Clinical
SZALVIJBUOXUFB 9.0 IC50 2
TWUDJPWCVJDVTM 8.7 IC50 26
CQCHOVDIAHVBMQ 8.7 IC50 26
OCXSSYNPSCOWLL 8.7 IC50 2
UNDRZULXNGGEMB 8.7 IC50 2
ZMRQKZANSRISRS 8.7 IC50 3
LQNBSHGSEOTYDZ 8.6 IC50 26
JWUFFURPSKRHTA 8.5 IC50 2
TYXGRJPOMQEXJV 8.5 IC50 26
YOXMEVDONXENBC 8.5 IC50 2
GTVKXVAXHKIMQX 8.5 IC50 26
ZMRQKZANSRISRS 8.4 IC50 3
YOOPYOPIAKCHQH 8.3 IC50 2
HACCLYCGUNUBJY 8.2 IC50 26
FRGPFJVINLDQIJ 8.2 IC50 26
CMKXTNFXBYWXGN 8.2 IC50 2
JWZPZXKJEUAZFV 8.2 IC50 26
MFCDBQIDJOCFDS 8.2 IC50 2
RIAAESBLPRZGAK 8.2 IC50 26
AJCGCPQKWYQPNQ 8.1 IC50 26
DAMJJTRLEZYXQM 8.1 IC50 26
QUYJROSEXGBONG 8.1 IC50 26
XCEJVZUIMKOKDS 8.1 IC50 2
OXIUFIQCDNTAED 8.1 IC50 26
YEOAYGDVMJPHGG 8.0 IC50 26
OSYITGFTDTWGJW 8.0 IC50 26
UGCISYLUHGKJKT 8.0 IC50 26
SRGBARMXFGWMTF 7.9 IC50 26
CNCRGRBWUATVCP 7.8 IC50 26
YZIYDQGNWSHQSD 7.8 IC50 26
ZMYGBEMRHGJETO 7.8 IC50 26
NOCIOWGNSBLDHC 7.8 IC50 26
NWSFHJWTWBRJFA 7.8 IC50 26
AYXYPKUFHZROOJ 7.7 Ki 2
ZTKAJVXFDWQBSJ 7.7 IC50 3
XCLYWDHZGKKXTL 7.7 IC50 2
CLSLOWKHEUDMRP 7.7 IC50 26
PSRVKIMUQGXDRE 7.7 IC50 2
AYXYPKUFHZROOJ 7.6 IC50 3
ZTNBOUBFOFURTR 7.6 IC50 26
INGBKPUFSDYYRV 7.6 IC50 2
PTYOAOCUXNHRIN 7.6 IC50 2
BDMBSHGVIWYMFZ 7.6 IC50 26
BDZDJFPQRUGPOF 7.5 IC50 26
BVNRYPXFJUABAB 7.5 IC50 26
UIAGMCDKSXEBJQ 7.5 IC50 4
NRQIYYZXZYUWFB 7.5 IC50 26
VLKBVXIFTQLGCO 7.5 IC50 26
MVUOEDQURQKALH 7.5 IC50 26
PSVKDIGKMXLUQF 7.5 IC50 26
2D structure