Target Details
| UniProt AC | P53985 |
|---|---|
| Gene Symbol | SLC16A1 |
| Protein Name | Monocarboxylate transporter 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07690 (MFS_1) |
Summary
- Multi-target molecules 41
- Clinical molecules 0
- Avg pChEMBL 7.27
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (41)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GOSZMIDOMHVHDD
|
10.1 | Ki | 2 | — | |
SJZYZYMKFRJDEE
|
9.6 | Ki | 2 | — | |
FPZKMOBZAQYAOC
|
9.4 | Ki | 2 | — | |
QFJAWVIERUMTED
|
9.0 | Ki | 2 | — | |
ISIVOJWVBJIOFM
|
8.9 | Ki | 2 | — | |
PRNXOFBDXNTIFG
|
8.8 | Kd | 3 | — | |
UHNVWCCKBJDIGZ
|
8.5 | Ki | 2 | — | |
JOFQERPJMGKMMX
|
8.3 | Ki | 2 | — | |
OOKBWQIMMUTDEE
|
8.1 | IC50 | 2 | — | |
KLVPSHRCXIALKY
|
7.9 | Ki | 2 | — | |
ZCCPLJOKGAACRT
|
7.3 | Kd | 599 | — | |
GWRCGDREYBGGOB
|
7.3 | IC50 | 2 | — | |
JKSRDKKNSRKQBO
|
7.3 | IC50 | 3 | — | |
OWAJCGGSUQXKSU
|
7.3 | IC50 | 2 | — | |
FVIJIRCHSMDMJH
|
7.2 | Ki | 2 | — | |
XTKDQPFUOFAMRL
|
7.2 | IC50 | 2 | — | |
RAJPEVIHJCKTGX
|
7.1 | IC50 | 2 | — | |
AMBDDVHEOJZXJJ
|
7.0 | IC50 | 3 | — | |
PPYZGAFFTAKWEP
|
7.0 | IC50 | 3 | — | |
DJOMFUVHYJYBLP
|
7.0 | IC50 | 2 | — | |
JGBAQQPRYIWBBM
|
7.0 | IC50 | 2 | — | |
SXTVAMOLTIPBMD
|
7.0 | IC50 | 2 | — | |
KBBKSCWNTBRVIG
|
6.8 | IC50 | 2 | — | |
LONCIMGLEVRXRB
|
6.8 | IC50 | 2 | — | |
RTWRTPIGKUMZKL
|
6.8 | IC50 | 2 | — | |
QBORYSJTYYBZDK
|
6.7 | IC50 | 2 | — | |
YWAWTBJHCYHBMP
|
6.7 | IC50 | 3 | — | |
ZRXMBBHQLHYREE
|
6.7 | IC50 | 3 | — | |
LUDYZNVCPGSFNX
|
6.7 | IC50 | 2 | — | |
UBHYMOUAWIJFLD
|
6.6 | IC50 | 2 | — | |
YKNHVSZOKRRXNB
|
6.6 | IC50 | 2 | — | |
BEHYBUQUZGAMAX
|
6.5 | IC50 | 3 | — | |
IRHLEONWFSXRDD
|
6.5 | IC50 | 3 | — | |
RUFWXTRLNGUAJT
|
6.5 | IC50 | 3 | — | |
RZGBMPZXWLXWJO
|
6.4 | IC50 | 3 | — | |
OMJMCBRZEPPIAA
|
6.4 | IC50 | 3 | — | |
SGFRVEMOPYHHFG
|
6.4 | IC50 | 3 | — | |
GMVVYVHASOEGGH
|
6.3 | IC50 | 2 | — | |
HMGBBPKGJHXSQG
|
6.3 | IC50 | 2 | — | |
FBBHOORHLONXEV
|
6.2 | IC50 | 2 | — | |
WHCPTFFIERCDSB
|
6.1 | IC50 | 2 | — |