Target Details
| UniProt AC | P53779 |
|---|---|
| Gene Symbol | MAPK10 |
| Protein Name | Mitogen-activated protein kinase 10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 625
- Clinical molecules 259
- Avg pChEMBL 7.25
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (625)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GBKQNVNYZATRQE
|
7.0 | IC50 | 2 | Yes | |
NRJKIOCCERLIDG
|
7.0 | Kd | 6 | — | |
QVEWXFMWNGGSAH
|
7.0 | IC50 | 3 | Yes | |
BCNMJLRKWYKBBZ
|
7.0 | IC50 | 4 | — | |
ASGMFNBUXDJWJJ
|
7.0 | IC50 | 8 | — | |
HGCVWICUBZDORS
|
7.0 | IC50 | 2 | — | |
HXZDICYKFAOZLE
|
7.0 | IC50 | 6 | Yes | |
IBSOKDKEFQOSIY
|
7.0 | IC50 | 2 | Yes | |
IOBZIJYYPWNRQU
|
7.0 | IC50 | 3 | Yes | |
QYYMQRVJYZKVBE
|
7.0 | IC50 | 2 | — | |
RXFZUHJHYNKIJF
|
7.0 | IC50 | 2 | Yes | |
SZHHSFHOIDCNLD
|
7.0 | Kd | 6 | — | |
SZHHSFHOIDCNLD
|
7.0 | Kd | 3 | — | |
YPAADIPEHKVUEJ
|
7.0 | IC50 | 2 | Yes | |
AHYIIKWTYMCFNB
|
7.0 | IC50 | 3 | — | |
PKNYJVSQHRVGTB
|
7.0 | IC50 | 2 | — | |
YTPKEJXVUUNXRA
|
7.0 | IC50 | 4 | Yes | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 213 | — | |
JUCZVVOFLZHKJP
|
7.0 | IC50 | 2 | Yes | |
KEJPODFMUKBEAK
|
7.0 | IC50 | 3 | Yes | |
MHEZQXUHNPRCFQ
|
7.0 | IC50 | 2 | Yes | |
YKQSOUXCRZONQQ
|
7.0 | IC50 | 3 | Yes | |
DKZYXHCYPUVGAF
|
7.0 | Kd | 112 | — | |
CUDZNCZDKGCXRX
|
6.9 | IC50 | 2 | — | |
FEENLVZHRIAWGM
|
6.9 | IC50 | 2 | — | |
JFCLFMVVHSGPDK
|
6.9 | IC50 | 3 | — | |
JSQNZBQJTQNCFK
|
6.9 | IC50 | 7 | — | |
LTKLQMAKAFTREX
|
6.9 | IC50 | 2 | Yes | |
RJVBVUWFYMRHRI
|
6.9 | IC50 | 4 | Yes | |
YAJKXICRGUNBDU
|
6.9 | IC50 | 2 | — | |
QLDFAHVPALXKAU
|
6.9 | IC50 | 2 | — | |
VYQHPOVDIRILEA
|
6.9 | IC50 | 3 | Yes | |
CDHZIFBQYVOWNY
|
6.9 | IC50 | 3 | — | |
HZTYDQRUAWIZRE
|
6.9 | Kd | 40 | Yes | |
QUBFVDVWHOIYRD
|
6.9 | IC50 | 2 | — | |
UCPDQFHGSDFSKX
|
6.9 | IC50 | 2 | Yes | |
VLMWLALTUHMVKC
|
6.9 | IC50 | 2 | — | |
VQAHFLPDFJAHTG
|
6.9 | IC50 | 2 | Yes | |
XMMMRYGZMVXRBI
|
6.9 | IC50 | 2 | — | |
BYCDZWGPIIHWFV
|
6.9 | IC50 | 2 | Yes | |
GTIQIAGCTCXGCN
|
6.9 | IC50 | 2 | — | |
JCLKKRZMUZBICB
|
6.9 | IC50 | 2 | — | |
HMLQTEJXWLWZJQ
|
6.9 | IC50 | 2 | — | |
CEJFYMKXALJHTD
|
6.8 | IC50 | 2 | Yes | |
JSGWWFGFBLUWSD
|
6.8 | IC50 | 2 | Yes | |
LJWSUGUZCIJVRS
|
6.8 | IC50 | 2 | Yes | |
VHYFUPDFEUQXIH
|
6.8 | IC50 | 2 | Yes | |
DVRSTRMZTAPMKO
|
6.8 | IC50 | 10 | Yes | |
HQBDXBBDGWHRLC
|
6.8 | IC50 | 3 | Yes |