Target Details
| UniProt AC | P53779 |
|---|---|
| Gene Symbol | MAPK10 |
| Protein Name | Mitogen-activated protein kinase 10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 625
- Clinical molecules 259
- Avg pChEMBL 7.25
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (625)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JRCVTCDIBTUNEL
|
7.2 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
7.2 | Kd | 231 | Yes | |
WQYDASORCSDVNY
|
7.2 | IC50 | 2 | — | |
AVLYNJZZQYEFEA
|
7.2 | IC50 | 8 | Yes | |
CUABCZMVBDQUGO
|
7.2 | IC50 | 2 | Yes | |
KORISVSXBGATCA
|
7.2 | IC50 | 2 | — | |
NUEDKDFHLPVYRY
|
7.2 | IC50 | 2 | Yes | |
OOOZOACKEXWXQJ
|
7.2 | IC50 | 3 | Yes | |
PXOJJCCSYAVCPK
|
7.2 | IC50 | 3 | Yes | |
UHNHUQMERWMFSO
|
7.2 | IC50 | 2 | Yes | |
GFABXPYEGAFBKF
|
7.2 | IC50 | 2 | — | |
PHDVAWAUKMHEJM
|
7.2 | IC50 | 3 | Yes | |
RCYPVQCPYKNSTG
|
7.2 | IC50 | 7 | — | |
STRBDWNAMGZLQF
|
7.1 | IC50 | 2 | Yes | |
UIRLFLOVKAOFEX
|
7.1 | Ki | 3 | Yes | |
WVXNSAVVKYZVOE
|
7.1 | Kd | 92 | — | |
RXDOUBRAWQLAGH
|
7.1 | IC50 | 3 | — | |
UVMRYWDKSNEROE
|
7.1 | IC50 | 2 | — | |
BTJOSZCOBPWUOW
|
7.1 | Kd | 3 | — | |
BGGSTZPBQKGLOJ
|
7.1 | IC50 | 3 | Yes | |
IVUHAOSDDKKRTF
|
7.1 | IC50 | 2 | — | |
JKCOWGOVZGAWTE
|
7.1 | IC50 | 2 | Yes | |
JVSLZGKNRZILCQ
|
7.1 | IC50 | 2 | — | |
NCUDSKLYBDQTIW
|
7.1 | IC50 | 2 | — | |
PZILHQVGAVFRNS
|
7.1 | IC50 | 2 | — | |
VFBUSLHLJVREKP
|
7.1 | IC50 | 2 | Yes | |
WEKXWKLEXYHQPV
|
7.1 | IC50 | 2 | — | |
YPUXXNJBUOZMOQ
|
7.1 | IC50 | 3 | Yes | |
YRFPTZPAVDAEDW
|
7.1 | IC50 | 2 | Yes | |
ZNXYLXPOVFQCEW
|
7.1 | IC50 | 2 | — | |
FPOJVFPVFJTSDR
|
7.1 | IC50 | 3 | — | |
VFDMQZQCLWTEJN
|
7.1 | IC50 | 3 | Yes | |
YMRWBKJYJJXFPZ
|
7.1 | IC50 | 2 | — | |
FVONQZQMUHLATI
|
7.1 | IC50 | 3 | — | |
MVCOAUNKQVWQHZ
|
7.1 | Kd | 54 | Yes | |
SVIILPGBQTUQPJ
|
7.1 | IC50 | 2 | — | |
BCIAPPMPZKEHOE
|
7.1 | IC50 | 3 | — | |
LCBNUBGZQBBNPG
|
7.1 | IC50 | 2 | Yes | |
UNWYPVDZMQJENJ
|
7.1 | IC50 | 2 | Yes | |
ZECOHPFWGOCWLO
|
7.1 | IC50 | 5 | — | |
ACPOUJIDANTYHO
|
7.0 | IC50 | 17 | Yes | |
CEFHLBGJHWUOBZ
|
7.0 | Ki | 3 | — | |
HGQHCYUSXPTRID
|
7.0 | IC50 | 4 | Yes | |
HJJSEANNATVFNW
|
7.0 | IC50 | 4 | — | |
KRIUNPBAQZGFQA
|
7.0 | IC50 | 76 | — | |
SLMJDPXFWRYMLU
|
7.0 | IC50 | 3 | — | |
TWTIIHVYOGLKME
|
7.0 | Ki | 3 | Yes | |
USOOZXUJZKQXCC
|
7.0 | IC50 | 3 | — | |
DQAXOJBNTQVNHJ
|
7.0 | IC50 | 2 | — | |
JPTYCOMKVYISJL
|
7.0 | IC50 | 2 | Yes |