Target Details
| UniProt AC | P53779 |
|---|---|
| Gene Symbol | MAPK10 |
| Protein Name | Mitogen-activated protein kinase 10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 625
- Clinical molecules 259
- Avg pChEMBL 7.25
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (625)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CCDFASODNLEBEJ
|
6.6 | IC50 | 3 | — | |
XCPPIJCBCWUBNT
|
6.6 | IC50 | 3 | — | |
HYYRJELYMNIRGB
|
6.6 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
6.6 | Kd | 103 | — | |
IEZJTLFFNLOEKV
|
6.6 | IC50 | 3 | — | |
MSNLSSCFMUKCNV
|
6.6 | IC50 | 3 | — | |
RHLSCLBSPZIGFS
|
6.6 | IC50 | 3 | Yes | |
SGWLRDAOCLITOM
|
6.6 | IC50 | 7 | — | |
VUQJMYORHRVTLM
|
6.6 | IC50 | 3 | — | |
ZVDDPXIWKBBCQE
|
6.6 | IC50 | 3 | Yes | |
GLFSGNWAZDGYBV
|
6.6 | IC50 | 2 | Yes | |
NHSDXYBXQGQSRA
|
6.6 | IC50 | 3 | — | |
OSVUGUHRKMMBSE
|
6.6 | Kd | 170 | — | |
KTBZRPANEUUZDW
|
6.6 | IC50 | 2 | — | |
MZDKLVOWGIOKTN
|
6.6 | Ki | 80 | — | |
NEBNIXUGANAKDR
|
6.6 | IC50 | 2 | Yes | |
RDNOLDWOMGZBPI
|
6.6 | IC50 | 8 | Yes | |
RSBSYGXBCWDUEI
|
6.6 | IC50 | 2 | Yes | |
UDOITUAULPBVSE
|
6.6 | IC50 | 3 | Yes | |
XYVNGBDEDFMYEK
|
6.6 | IC50 | 2 | Yes | |
ZMFVICCTJZQVDM
|
6.6 | IC50 | 3 | — | |
QWWPWWKJOUHOAP
|
6.6 | IC50 | 2 | — | |
MZFRCQRBHBNGFV
|
6.6 | IC50 | 2 | Yes | |
YPXNJMUSTWLKRM
|
6.6 | IC50 | 2 | Yes | |
BKLYUVKUMMLBIJ
|
6.6 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
6.6 | Kd | 165 | Yes | |
PMNWPSRSXHKOQI
|
6.6 | Kd | 3 | — | |
DGYKSZOQVJDTRZ
|
6.5 | Kd | 2 | — | |
ZYPRSWQPKLBUQM
|
6.5 | IC50 | 3 | Yes | |
PPHUYGGBTOACGL
|
6.5 | IC50 | 2 | Yes | |
QVMKLKBODZHJDK
|
6.5 | IC50 | 2 | — | |
SSWFFPALFQMQLE
|
6.5 | IC50 | 3 | — | |
PRFQGCBPEYPZAY
|
6.5 | IC50 | 3 | — | |
HHAPAAFKKUAWAI
|
6.5 | IC50 | 5 | — | |
INGLARCWUNLRGV
|
6.5 | IC50 | 2 | Yes | |
JTVHPFGRRUKYMR
|
6.5 | IC50 | 3 | Yes | |
KDKUVYLMPJIGKA
|
6.5 | Ki | 91 | Yes | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
UPOMRTKHZCWMBW
|
6.5 | IC50 | 2 | — | |
IQCBETQVXZDQOC
|
6.5 | IC50 | 2 | — | |
LRMJMUNRVWCGNU
|
6.5 | IC50 | 2 | Yes | |
SIBBXUMRESEGRS
|
6.5 | IC50 | 3 | — | |
WYBUPBYFJYBWQP
|
6.5 | IC50 | 2 | — | |
DZCSIYOZJRMQKN
|
6.5 | IC50 | 2 | Yes | |
HPQZTEVMVAVGJO
|
6.5 | Kd | 5 | — | |
BDHQTRQDQKVEIM
|
6.5 | IC50 | 3 | Yes | |
HZYXRWDUVNONMO
|
6.5 | IC50 | 2 | — | |
IUDPPAXWQBHYHO
|
6.5 | IC50 | 2 | — | |
LZFPDJIWDHUHJG
|
6.5 | IC50 | 3 | — | |
MKUCYQPSROSPGD
|
6.5 | IC50 | 4 | Yes |