Target Details
| UniProt AC | P53708 |
|---|---|
| Gene Symbol | ITGA8 |
| Protein Name | Integrin alpha-8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) PF00357 (Integrin_alpha) |
Summary
- Multi-target molecules 21
- Clinical molecules 0
- Avg pChEMBL 8.8
KEGG Pathways (11)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
Associated Diseases (1)
Active Molecules (21)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SHRSEUHJTZQLRO
|
9.4 | IC50 | 8 | — | |
BQYBIJDRTDZCAJ
|
9.3 | IC50 | 8 | — | |
JXVVEFIKDDVLOS
|
9.3 | IC50 | 8 | — | |
QTBFGJFGHGTDRF
|
9.3 | IC50 | 8 | — | |
MFCABRSSOZYCRL
|
9.2 | IC50 | 8 | — | |
PEFBVOAICYLSAF
|
9.2 | IC50 | 8 | — | |
RTYLRDWEJUNBLU
|
9.2 | IC50 | 8 | — | |
YPAMHQMVIMQKOR
|
9.2 | IC50 | 8 | — | |
OBOJFQICXTYCRY
|
9.2 | IC50 | 8 | — | |
XRXSSPOFDFFALK
|
9.2 | IC50 | 8 | — | |
UCBYYQWMMNUSGH
|
9.1 | IC50 | 8 | — | |
GDEQKRGKHZOXGD
|
9.1 | IC50 | 8 | — | |
HIKDGFUZLZJZCB
|
9.1 | IC50 | 8 | — | |
QLBXWVBTUGYSGI
|
9.0 | IC50 | 8 | — | |
ZAMKDPACDNUZPJ
|
8.9 | IC50 | 8 | — | |
BWAUVRFZNDRMLY
|
8.9 | IC50 | 8 | — | |
CJRDXSVCUSRJDR
|
8.8 | IC50 | 8 | — | |
CJFKBQRLRONQOT
|
8.5 | IC50 | 7 | — | |
RBJQMIIPTLTYFP
|
7.4 | IC50 | 8 | — | |
ILKRHUYCJMCBRQ
|
7.2 | IC50 | 8 | — | |
XWMGBLCMRLASDS
|
6.4 | IC50 | 8 | — |