Target Details
| UniProt AC | P53667 |
|---|---|
| Gene Symbol | LIMK1 |
| Protein Name | LIM domain kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00412 (LIM) PF00595 (PDZ) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 364
- Clinical molecules 14
- Avg pChEMBL 7.01
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (364)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KWRXWPRFIUJQBP
|
6.0 | Ki | 25 | — | |
KWSZYBNXNYRQCC
|
6.0 | Ki | 21 | — | |
LNIDFQVRZCDVBI
|
6.0 | Ki | 16 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NLUPJKQOKWBWFC
|
6.0 | Ki | 69 | — | |
OVKIYZXGCCAIJG
|
6.0 | Ki | 6 | — | |
SXUFGUQQFYCNHW
|
6.0 | IC50 | 2 | — | |
UCLBDUZAAUTHBW
|
6.0 | Ki | 4 | — | |
UCOWZARZLHNDKP
|
6.0 | Ki | 8 | — | |
ULHGAQSVFPOUDY
|
6.0 | Ki | 43 | — | |
VAARYSWULJUGST
|
6.0 | Kd | 119 | Yes | |
XNEPVLVYFUGJLF
|
6.0 | Ki | 27 | — | |
ZLHFILGSQDJULK
|
6.0 | Ki | 37 | Yes | |
ZWENVGPTFUGBBT
|
6.0 | Ki | 2 | — |